SCHEMBL8720079

SCHEMBL8720079

CCC(C(=O)O)c1cc(C)[nH]n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 7/20 0.46
DAO P14920 1/20 0.46
HCAR3 P49019 3/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CCNA1 P78396 1/20 0.36
AKR1C3 P42330 6/20 0.36
AKR1C2 P52895 6/20 0.36
AKR1C1 Q04828 1/20 0.36
PTGS1 P23219 1/20 0.36
ALPL P05186 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1206525 0.72 HCAR2 (0.35) HCAR2DAOHCAR3ALPLL3MBTL1
SCHEMBL1531197 0.69 HCAR2 (0.42) HCAR2DAOHCAR3AKR1C3AKR1C2
SCHEMBL16619099 0.68 BRD4 (0.39) HCAR2DAOCCNA2CDK2CCNA1
SCHEMBL16619580 0.68 HCAR2 (0.32) HCAR2DAOALPLL3MBTL1
SCHEMBL26775764 0.68 CYP1A2 (0.34) HCAR2DAOL3MBTL1
SCHEMBL3740712 0.68 AKR1C3 (0.40) AKR1C3AKR1C2AKR1C1PTGS1
SCHEMBL15218944 0.67 HCAR2 (0.62) HCAR2DAOHCAR3ALPLL3MBTL1
SCHEMBL10761856 0.67 AKR1C3 (0.36) HCAR3AKR1C3AKR1C2AKR1C1PTGS1
SCHEMBL31554349 0.67 AKR1C3 (0.33) AKR1C3AKR1C2AKR1C1PTGS1
SCHEMBL804646 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0879234-A1 1-PYRAZOL-3-YL-ETHYL-4-INDOL-3-YL-PIPERIDINE USED AS MEDICINE ACTING ON THE CENTRAL NERVOUS SYSTEM MERCK PATENT GmbH (DE) 1998-11-25 EP disclosed
WO-1997027186-A1 1-PYRAZOL-3-YL-ETHYL-4-INDOL-3-YL-PIPERIDINE USED AS MEDICINE ACTING ON THE CENTRAL NERVOUS SYSTEM MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-07-31 WO disclosed