SCHEMBL8739768

SCHEMBL8739768

O=C(Cn1nc(-c2ccc(Cl)cc2)n(Cc2ccccc2F)c1=O)NCc1c(C(F)F)cccc1C(F)(F)F

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 18/20 0.60
AVPR1A P37288 18/20 0.60
NR1H2 P55055 1/20 0.42
NR1H3 Q13133 1/20 0.42
CNR1 P21554 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8235588 0.93 AVPR2 (0.59) AVPR2AVPR1ANR1H2NR1H3CNR1
SCHEMBL8235014 0.92 AVPR2 (0.58) AVPR2AVPR1ANR1H2NR1H3CNR1
SCHEMBL8227362 0.88 AVPR2 (0.60) AVPR2AVPR1ANR1H2NR1H3CNR1
SCHEMBL8232587 0.87 AVPR2 (0.58) AVPR2AVPR1ANR1H2NR1H3CNR1
SCHEMBL8232897 0.87 AVPR2 (0.57) AVPR2AVPR1ANR1H2NR1H3CNR1
SCHEMBL8232603 0.87 AVPR2 (0.57) AVPR2AVPR1ANR1H2NR1H3CNR1
SCHEMBL8234745 0.85 AVPR2 (0.53) AVPR2AVPR1ACNR1
SCHEMBL19244834 0.85 AVPR2 (0.61) AVPR2AVPR1ANR1H2NR1H3
SCHEMBL19244833 0.84 AVPR2 (0.59) AVPR2AVPR1ANR1H2NR1H3
SCHEMBL8227858 0.84 AVPR2 (0.68) AVPR2AVPR1ACNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027096-B1 SUBSTITUTED ARYLIMIDAZ0L0NE AND TRIAZ0L0NE AS INHIBITORS OF VASOPRESSIN RECEPTORS Bayer Pharma AG (DE) 2012-05-23 EP disclosed