SCHEMBL87417

SCHEMBL87417

Cc1cc(CNC(=O)c2nc3n(c(=O)c2O)CC2CCC3(N(C)C(=O)C(=O)N3CCCC3)CC2)ccc1F

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.44
KCNH2 Q12809 1/20 0.41
MMP13 P45452 8/20 0.35
ALDH1A1 P00352 3/20 0.33
LMNA P02545 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
CALCA P06881 2/20 0.33
GAA P10253 1/20 0.32
MMP10 P09238 3/20 0.32
MMP8 P22894 3/20 0.32
MMP9 P14780 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL52304 0.93 CYP2C9 (0.40) CYP2C9KCNH2MMP13ALDH1A1LMNA
SCHEMBL52108 0.91 CYP2C9 (0.54) CYP2C9KCNH2ALDH1A1LMNAMAPT
SCHEMBL51612 0.91 CYP2C9 (0.47) CYP2C9KCNH2MMP13ALDH1A1LMNA
SCHEMBL53150 0.86 CYP2C9 (0.39) CYP2C9KCNH2MMP13MMP10MMP8
SCHEMBL53118 0.85 CYP2C9 (0.39) CYP2C9KCNH2MMP13ALDH1A1KDM4E
SCHEMBL10144275 0.85 CYP2C9 (0.49) CYP2C9KCNH2CALCAGAA
SCHEMBL52672 0.85 CYP2C9 (0.48) CYP2C9KCNH2MMP13ALDH1A1LMNA
SCHEMBL418770 0.84 CYP2C9 (0.49) CYP2C9KCNH2LMNACALCA
SCHEMBL9904916 0.84 CYP2C9 (0.40) CYP2C9KCNH2MMP13ALDH1A1LMNA
SCHEMBL52047 0.83 CYP2C9 (0.49) CYP2C9KCNH2LMNAMAPTCALCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129398-B2 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-06 US disclosed
US-20090253677-A1 HIV Integrase Inhibitors BRISTOL-MYERS SQUIBB COMPANY 2009-10-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090253677-A1 HIV Integrase Inhibitors DNTT, POLB, UNG CYP2C9 602/4885KCNH2 3969/4885MMP13 4137/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.