SCHEMBL8746808

SCHEMBL8746808

O=C=Nc1ccc(C(Cl)(Cl)Cl)cc1Cl

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
TDP1 Q9NUW8 2/20 0.40
MAPK1 P28482 1/20 0.40
CYP3A4 P08684 3/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
TRPA1 O75762 1/20 0.34
GABRA1 P14867 1/20 0.32
GABRB2 P47870 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11872628 0.89 TDP1 (0.40) TSHRTDP1MAPK1CYP3A4ALDH1A1
SCHEMBL11872782 0.86 TDP1 (0.38) TSHRTDP1MAPK1CYP3A4ALDH1A1
SCHEMBL10791997 0.85 TSHR (0.50) TSHRTDP1MAPK1CYP3A4ALDH1A1
SCHEMBL3960923 0.84 TDP1 (0.39) TSHRTDP1MAPK1CYP3A4ALDH1A1
SCHEMBL162605 0.84 PDE2A (0.41) TSHRTDP1MAPK1CYP3A4ALDH1A1
SCHEMBL29648890 0.84 PDE2A (0.41) TSHRTDP1MAPK1CYP3A4ALDH1A1
SCHEMBL11782324 0.80 TSHR (0.35) TSHRTDP1MAPK1CYP3A4ALDH1A1
SCHEMBL27701883 0.80 TDP1 (0.36) TDP1MAPK1CYP3A4ALDH1A1HPGD
SCHEMBL8746797 0.79 TSHR (0.45) TSHRTDP1MAPK1GABRA1GABRB2
SCHEMBL29565739 0.76 CYP3A4 (0.53) TSHRTDP1MAPK1CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107098817-A 2,6- of one kind dichlor-4-trifluoromethyl anilines lead to chlorine production technology 江苏托球农化股份有限公司 2017-08-29 CN disclosed
EP-0639556-B1 Process for the preparation of trifluoromethylanilines HOECHST AG (DE) 1997-03-05 EP disclosed
US-5471002-A Process for preparing trifluoromethylanilines CLARIANT PRODUKTE (DEUTSCHLAND) GMBH (DE) 1995-11-28 US disclosed
EP-0639556-A1 Process for the preparation of trifluoromethylanilines HOECHST AKTIENGESELLSCHAFT (DE) 1995-02-22 EP disclosed
US-4950813-A Preparation of substituted benzotrichlorides BAYER AKTIENGESELLSCHAFT (DE) 1990-08-21 US disclosed
EP-0306804-A2 Process for the preparation of substituted benzyl trichlorides BAYER AG (DE) 1989-03-15 EP disclosed
US-4748277-A FLUORINATION AND HYDROLYSIS OF TRIHALOMETHYLPHENYL ISOCYANATE RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1988-05-31 US disclosed
EP-0012435-A2 Isoxazole derivatives, process for their preparation, medicines containing them and intermediates required in this process HOECHST AKTIENGESELLSCHAFT (DE) 1980-06-25 EP disclosed