SCHEMBL8752192

SCHEMBL8752192

C=CC(Cn1cnc2c(Cl)nc(N)nc21)OC(C(C)C)(C(C)C)P(=O)(O)O

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 4/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC4 P56524 1/20 0.42
HSP90AB1 P08238 13/20 0.41
HSP90AA1 P07900 12/20 0.41
HSP90B1 P14625 1/20 0.39
TRAP1 Q12931 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
FDPS P14324 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8752200 1.00 HDAC6 (0.42) HDAC6HDAC1HDAC4HSP90AB1HSP90AA1
SCHEMBL9176450 0.87 HDAC6 (0.46) HDAC6HDAC1HDAC4HSP90AB1HSP90AA1
SCHEMBL6004037 0.82 HSP90AB1 (0.42) HDAC6HDAC1HDAC4HSP90AB1HSP90AA1
SCHEMBL6004500 0.82 HSP90AB1 (0.42) HDAC6HDAC1HDAC4HSP90AB1HSP90AA1
SCHEMBL8752184 0.78 HSP90AB1 (0.43) HDAC6HDAC1HDAC4HSP90AB1HSP90AA1
SCHEMBL6004535 0.78 HSP90AB1 (0.41) HDAC6HDAC1HDAC4HSP90AB1HSP90AA1
SCHEMBL8752233 0.78 HSP90AB1 (0.43) HDAC6HDAC1HDAC4HSP90AB1HSP90AA1
SCHEMBL17254507 0.77 HSP90AB1 (0.46) HDAC6HDAC1HDAC4HSP90AB1HSP90AA1
SCHEMBL14244312 0.77 HSP90AB1 (0.46) HDAC6HDAC1HDAC4HSP90AB1HSP90AA1
SCHEMBL6002747 0.77 HSP90AB1 (0.42) HDAC6HDAC1HDAC4HSP90AB1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696263-A Antiviral acyclic phosphonomethoxyalkylsubstituted alkenyl and alkynyl purine and pyrimidine derivatives INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 1997-12-09 US disclosed
EP-0630381-B1 ANTIVIRAL ACYCLIC PHOSPHONOMETHOXYALKYL SUBSTITUTED, ALKENYL AND ALKYNYL PURINE AND PYRIMIDINE DERIVATIVES ACAD OF SCIENCE CZECH REPUBLIC (CZ) 1997-04-09 EP disclosed
WO-1993007157-A1 ANTIVIRAL ACYCLIC PHOSPHONOMETHOXYALKYL SUBSTITUTED, ALKENYL AND ALKYNYL PURINE AND PYRIMIDINE DERIVATIVES INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OFTHE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 1993-04-15 WO disclosed