SCHEMBL8765956

SCHEMBL8765956

CSC1(SC)CCOc2ccc(C#Cc3ccc(CCO)cn3)cc21

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.35
RARA P10276 1/20 0.35
RARB P10826 1/20 0.35
RARG P13631 1/20 0.35
KMT2A Q03164 1/20 0.35
FFAR1 O14842 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35
ACACB O00763 4/20 0.34
CYP26A1 O43174 1/20 0.34
CHEK1 O14757 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL860638 0.92 CYP3A4 (0.36) CYP3A4RARARARBRARGKMT2A
SCHEMBL6670288 0.87 CYP26A1 (0.39) CYP3A4RARARARBRARGKMT2A
SCHEMBL6671545 0.83 CYP3A4 (0.42) CYP3A4RARARARBRARGKMT2A
SCHEMBL5485075 0.83 BACE1 (0.39) CYP3A4RARARARBRARGKMT2A
SCHEMBL180443 0.82 CYP3A4 (0.38) CYP3A4RARARARBRARGKMT2A
SCHEMBL1271404 0.81 CYP3A4 (0.54) CYP3A4RARARARBRARGKMT2A
SCHEMBL1078963 0.79 CYP3A4 (0.60) CYP3A4RARARARBRARGKMT2A
SCHEMBL28489810 0.79 GRM5 (0.50) CYP3A4RARARARBRARGKMT2A
SCHEMBL6665003 0.79 RARB (0.44) CYP3A4RARARARBRARGKMT2A
SCHEMBL20636822 0.77 CYP3A4 (0.41) CYP3A4RARARARBRARGKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785782-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1997-07-30 EP disclosed
WO-1996011686-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1996-04-25 WO disclosed