SCHEMBL8772678

SCHEMBL8772678

CCCN(C(=O)C(F)(F)F)c1ccc(I)cc1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 12/20 0.46
MEN1 O00255 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TP53 P04637 1/20 0.36
SERPINE1 P05121 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31211648 0.83 SMN1; SMN2 (0.59) MLYCDMEN1CYP3A4CYP2C9CYP2C19
SCHEMBL1312005 0.74 MAPT (0.44) MLYCDMEN1KMT2ASMN1; SMN2
SCHEMBL31211569 0.73 NPC1 (0.60) MLYCDMEN1CYP3A4CYP2C9CYP2C19
SCHEMBL31211559 0.72 NPC1 (0.62) MLYCDMEN1CYP3A4CYP2C9CYP2C19
SCHEMBL3270531 0.72 NPC1 (0.45) MLYCDMEN1KMT2ATP53
SCHEMBL11070556 0.72 NPC1 (0.48) MLYCDMEN1KMT2ATP53
SCHEMBL11562137 0.71 NPC1 (0.47) MLYCDTP53
SCHEMBL11559695 0.71 NPC1 (0.47) MLYCDTP53
SCHEMBL11561291 0.71 NPC1 (0.47) MLYCDTP53
SCHEMBL11063213 0.71 NPC1 (0.47) MLYCDTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691349-A ANTICHOLESTEROL AGENTS; ATHEROSCLEROSIS ZENECA LIMITED (GB) 1997-11-25 US disclosed
EP-0654032-B1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS ZENECA LTD (GB) 1997-10-15 EP disclosed
EP-0654032-A1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS. ZENECA LTD (GB) 1995-05-24 EP disclosed
WO-1994003451-A1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS ZENECA LIMITED (GB) 1994-02-17 WO disclosed