SCHEMBL8774900

SCHEMBL8774900

CCCOc1ccc(-c2ccc(-c3cnc(F)c(F)c3)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 6/20 0.46
CYP3A4 P08684 4/20 0.46
RAB9A P51151 7/20 0.46
NPC1 O15118 6/20 0.46
SMN1; SMN2 Q16637 5/20 0.46
ALDH1A1 P00352 3/20 0.46
MAPT P10636 1/20 0.46
RARA P10276 1/20 0.45
RARB P10826 1/20 0.45
CYP19A1 P11511 3/20 0.44
CYP2C9 P11712 3/20 0.44
CYP2C19 P33261 3/20 0.44
GRM5 P41594 1/20 0.44
ACACB O00763 1/20 0.43
ACACA Q13085 1/20 0.43
KDM4E B2RXH2 3/20 0.42
HSD17B10 Q99714 3/20 0.42
HPGD P15428 2/20 0.42
ALOX12 P18054 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774212 1.00 CYP2D6 (0.46) CYP2D6CYP3A4RAB9ANPC1SMN1; SMN2
SCHEMBL8774455 0.94 CYP2D6 (0.54) CYP2D6CYP3A4RAB9ANPC1SMN1; SMN2
SCHEMBL8774691 0.94 CYP2D6 (0.54) CYP2D6CYP3A4RAB9ANPC1SMN1; SMN2
SCHEMBL8774674 0.91 CYP2D6 (0.51) CYP2D6CYP3A4RAB9ANPC1SMN1; SMN2
SCHEMBL8774459 0.91 CYP2D6 (0.51) CYP2D6CYP3A4RAB9ANPC1SMN1; SMN2
SCHEMBL8774136 0.90 CYP2D6 (0.50) CYP2D6CYP3A4RAB9ANPC1SMN1; SMN2
SCHEMBL8774987 0.87 CHRNA7 (0.49) RAB9ANPC1ALDH1A1CYP19A1GRM5
SCHEMBL8774745 0.87 CHRNA7 (0.49) RAB9ANPC1ALDH1A1CYP19A1GRM5
SCHEMBL8774528 0.79 ACACB (0.42) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT
SCHEMBL8774590 0.79 ACACB (0.45) CYP2D6CYP3A4RAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed