SCHEMBL8775628

SCHEMBL8775628

O=C(Cc1ccccc1)NC1CCN(CCCC2(c3ccc(Cl)c(Cl)c3)COC(=O)N(Cc3ccccc3)C2)CC1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 10/20 0.54
TACR1 P25103 4/20 0.51
TACR2 P21452 3/20 0.51
TACR3 P29371 3/20 0.51
CCR5 P51681 3/20 0.49
CHRM1 P11229 2/20 0.46
CHRM2 P08172 1/20 0.46
CHRM4 P08173 1/20 0.46
CHRM5 P08912 1/20 0.46
DRD2 P14416 1/20 0.46
CHRM3 P20309 1/20 0.46
HTR2A P28223 1/20 0.46
ADRA1A P35348 1/20 0.46
HRH1 P35367 1/20 0.46
ADRA1B P35368 1/20 0.46
KCNH2 Q12809 1/20 0.46
MCHR1 Q99705 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4631187 0.85 TACR1 (0.52) TACR1TACR2TACR3CCR5
Hydrochloric Acid SCHEMBL7749174 0.85 TACR1 (0.52) TACR1TACR2TACR3CCR5
SCHEMBL4631687 0.84 TACR1 (0.51) TACR1TACR2TACR3CCR5
SCHEMBL4631231 0.82 TACR1 (0.53) TACR1TACR2TACR3CCR5CHRM2
SCHEMBL4631684 0.82 TACR1 (0.67) SIGMAR1TACR1TACR2TACR3CCR5
Hydrochloric Acid SCHEMBL7750128 0.82 TACR1 (0.52) TACR1TACR2TACR3CCR5CHRM2
SCHEMBL4630788 0.81 TACR3 (0.61) TACR1TACR2TACR3CCR5
Hydrochloric Acid SCHEMBL7750281 0.81 TACR1 (0.65) TACR1TACR2TACR3CCR5
Hydrochloric Acid SCHEMBL7750278 0.81 TACR1 (0.65) TACR1TACR2TACR3CCR5
Hydrochloric Acid SCHEMBL7750105 0.81 TACR3 (0.60) TACR1TACR2TACR3CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0807111-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI (FR) 1997-11-19 EP disclosed