SCHEMBL8775749

SCHEMBL8775749

C[C@@H]1Cc2cc(O)ccc2[C@@H]2[C@@H]1[C@@H]1CC[C@H](O)[C@@]1(C)C[C@@H]2O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 15/20 0.48
ESR2 Q92731 10/20 0.48
HSD17B10 Q99714 3/20 0.46
LMNA P02545 2/20 0.46
TSHR P16473 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HIF1A Q16665 1/20 0.46
SLC22A1 O15245 1/20 0.46
AKR1B10 O60218 1/20 0.46
SLC22A3 O75751 1/20 0.46
ABCB11 O95342 1/20 0.46
ESRRB O95718 1/20 0.46
ALDH1A1 P00352 1/20 0.46
NR3C1 P04150 1/20 0.46
SHBG P04278 1/20 0.46
PGR P06401 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14558087 0.92 ESR1 (0.48) ESR1ESR2HSD17B10LMNATSHR
SCHEMBL24103209 0.92 ESR1 (0.48) ESR1ESR2HSD17B10LMNATSHR
SCHEMBL24103208 0.92 ESR1 (0.48) ESR1ESR2HSD17B10LMNATSHR
SCHEMBL24102478 0.92 ESR1 (0.48) ESR1ESR2HSD17B10LMNATSHR
SCHEMBL6862563 0.87 ESR1 (0.45) ESR1ESR2HSD17B10LMNATSHR
SCHEMBL6862559 0.87 ESR1 (0.45) ESR1ESR2HSD17B10LMNATSHR
SCHEMBL24583080 0.83 ESR1 (0.63) ESR1ESR2HSD17B10LMNATSHR
SCHEMBL14569768 0.83 ESR1 (0.63) ESR1ESR2HSD17B10LMNATSHR
SCHEMBL24103217 0.83 ESR1 (0.63) ESR1ESR2HSD17B10LMNATSHR
SCHEMBL24103220 0.83 ESR1 (0.63) ESR1ESR2HSD17B10LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0719276-B1 ORALLY ACTIVE DERIVATIVES OF 1,3,5(10)-ESTRATRIENE US HEALTH (US) 1997-11-26 EP claimed
US-RE34136-E Morning-after contraceptives SRI INTERNATIONAL (US) 1992-12-01 US disclosed
EP-0227813-B1 11-BETA-NITRATE-SUBSTITUTED ESTRANES SRI INTERNATIONAL (US) 1991-10-02 EP disclosed
US-4859370-A 9 alpha, 11 beta-substituted and 11 beta-substituted estranes SRI INTERNATIONAL (US) 1989-08-22 US disclosed
US-4705783-A 9α, 11β-substituted and 11β-substituted estranes SRI INTERNATIONAL (US) 1987-11-10 US disclosed