SCHEMBL8775770

SCHEMBL8775770

CC(=O)Oc1ccc2c(c1)CC[C@H]1[C@@H]3CCC(=O)[C@@]3(C)C[C@H](O)[C@]21O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.56
STS P08842 5/20 0.51
ESR1 P03372 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
LMNA P02545 2/20 0.45
PGR P06401 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
AR P10275 1/20 0.45
CHRM1 P11229 1/20 0.45
TBXA2R P21731 1/20 0.45
ADRA1A P35348 1/20 0.45
OPRM1 P35372 1/20 0.45
SLC6A3 Q01959 1/20 0.45
ATM Q13315 1/20 0.45
CYP3A4 P08684 2/20 0.42
NR1H2 P55055 2/20 0.41
NR1H3 Q13133 2/20 0.41
HSD17B10 Q99714 2/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9746981 0.90 AKR1C3 (0.54) AKR1C3STSESR1SMN1; SMN2LMNA
SCHEMBL8775793 0.85 AKR1C3 (0.49) AKR1C3STSESR1SMN1; SMN2LMNA
SCHEMBL10770480 0.82 ESR1 (0.57) AKR1C3STSESR1LMNAPGR
SCHEMBL15295783 0.82 STS (0.57) AKR1C3STSESR1SMN1; SMN2LMNA
SCHEMBL10531124 0.82 AKR1C3 (0.52) AKR1C3STSESR1SMN1; SMN2LMNA
SCHEMBL9746143 0.80 ESR1 (0.46) AKR1C3STSESR1SMN1; SMN2LMNA
SCHEMBL9747077 0.77 STS (0.49) AKR1C3STSESR1SMN1; SMN2LMNA
SCHEMBL8776090 0.75 AKR1C3 (0.79) AKR1C3STSESR1SMN1; SMN2LMNA
SCHEMBL1688726 0.72 ESR1 (0.59) AKR1C3STSESR1SMN1; SMN2LMNA
SCHEMBL9747578 0.72 AKR1C3 (0.77) AKR1C3STSESR1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0719276-B1 ORALLY ACTIVE DERIVATIVES OF 1,3,5(10)-ESTRATRIENE US HEALTH (US) 1997-11-26 EP disclosed
US-RE34136-E Morning-after contraceptives SRI INTERNATIONAL (US) 1992-12-01 US disclosed
US-4859370-A 9 alpha, 11 beta-substituted and 11 beta-substituted estranes SRI INTERNATIONAL (US) 1989-08-22 US disclosed
US-4705783-A 9α, 11β-substituted and 11β-substituted estranes SRI INTERNATIONAL (US) 1987-11-10 US disclosed
WO-1987000175-A1 9alpha, 11beta-SUBSTITUTED AND 11beta-SUBSTITUTED ESTRANES SRI INTERNATIONAL (US) 1987-01-15 WO disclosed