SCHEMBL8787604

SCHEMBL8787604

COc1cc(CC=O)c(O)cc1OCCCCl

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 3/20 0.44
FDPS P14324 1/20 0.38
HTR2A P28223 2/20 0.38
PTPN1 P18031 3/20 0.36
PRSS1 P07477 3/20 0.35
ALDH1A1 P00352 3/20 0.35
MAPT P10636 3/20 0.35
KDM4E B2RXH2 2/20 0.35
MEN1 O00255 1/20 0.35
RECQL P46063 1/20 0.35
KMT2A Q03164 1/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
ALOX15 P16050 1/20 0.35
HTT P42858 2/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16445891 0.86 HMGCR (0.56) HMGCRPTPN1ALDH1A1MAPTKDM4E
SCHEMBL4764948 0.77 TAAR1 (0.44) HMGCRALDH1A1MAPTKDM4EMEN1
SCHEMBL3645037 0.77 HMGCR (0.42) HMGCRPTPN1ALDH1A1SMN1; SMN2
SCHEMBL6620053 0.77 PTGER4 (0.48) ALDH1A1MAPTKDM4EMEN1RECQL
SCHEMBL875687 0.77 HMGCR (0.44) HMGCRALDH1A1MAPTKDM4EMEN1
SCHEMBL16333910 0.75 HMGCR (0.65) HMGCRHTR2AHTT
SCHEMBL1766003 0.75 PPARA (0.54) FDPSALDH1A1MAPTKDM4EMEN1
SCHEMBL4774081 0.74 HMGCR (0.42) HMGCRHTR2AALDH1A1MAPTKDM4E
SCHEMBL3402738 0.74 EHMT2 (0.45)
SCHEMBL1545475 0.74 HTT (0.70) HMGCRALDH1A1MAPTKMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730452-A4 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST ROUSSEL PHARMA (US) 1997-03-19 EP disclosed
EP-0730452-A1 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST MARION ROUSSEL, Inc. (US) 1996-09-11 EP disclosed