SCHEMBL8794656

SCHEMBL8794656

CC1(C)C=C(c2ccc(C#N)nc2)c2cc(OC(F)(F)F)ccc2O1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.47
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
PGR P06401 1/20 0.35
SLC40A1 Q9NP59 1/20 0.35
ABL1 P00519 8/20 0.35
PGGT1B P53609 1/20 0.34
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34
KDM1A O60341 1/20 0.34
MAOB P27338 1/20 0.34
PDE10A Q9Y233 1/20 0.33
RARA P10276 2/20 0.33
RARB P10826 2/20 0.33
RARG P13631 2/20 0.33
GRM7 Q14831 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8795627 0.85 CHRM5 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8795372 0.85 PSEN1 (0.36) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8794401 0.83 PSEN1 (0.36) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8795556 0.81 DYRK1A (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8794852 0.80 CYP11B1 (0.43) ABL1SCN5ASCN9A
SCHEMBL8795654 0.79 ABL1 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8794555 0.78 ABL1 (0.36) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8794971 0.78 PSEN1 (0.35) TRPA1PSEN1PSEN2APH1BNCSTN
SCHEMBL8794576 0.74 CBFB (0.43) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8795589 0.72 PDE2A (0.42) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0485636-B1 INDOLE DERIVATIVE TORAY INDUSTRIES (JP) 1997-03-12 EP disclosed
EP-0735026-A1 Method for the production of isoquinoline derivatives and their use as intermediates in the preparation of indole derivatives TORAY INDUSTRIES, INC. (JP) 1996-10-02 EP disclosed
US-5539119-A MULTISTAGE FORMATION BY OXIDATION, REDUCING A CARBAMATE TO FORM AN ENAMINE, FORMING AN OXIDE TORAY INDUSTRIES, INC. (JP) 1996-07-23 US disclosed
EP-0485636-A1 INDOLE DERIVATIVE TORAY INDUSTRIES, INC. (JP) 1992-05-20 EP disclosed