SCHEMBL8799223

SCHEMBL8799223

O=C1NCC(CNC(c2ccccc2)c2ccccc2)c2c[nH]c3cccc1c23

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.41
PARP3 Q9Y6F1 1/20 0.32
MTOR P42345 1/20 0.31
RAB9A P51151 1/20 0.31
GRM7 Q14831 1/20 0.31
PIM1 P11309 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
JAK2 O60674 1/20 0.30
CYP3A4 P08684 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8798658 0.85 PARP1 (0.44) PARP1PIM1PIM2CYP3A4
Hydrochloric Acid SCHEMBL8800315 0.84 PARP1 (0.43) PARP1PIM1PIM2CYP3A4
SCHEMBL8798434 0.83 PARP1 (0.48) PARP1
Hydrochloric Acid SCHEMBL9484143 0.82 PARP1 (0.47) PARP1
Hydrochloric Acid SCHEMBL8800976 0.82 PARP1 (0.47) PARP1
Hydrochloric Acid SCHEMBL8801079 0.82 PARP1 (0.47) PARP1
SCHEMBL8798897 0.81 PARP1 (0.44) PARP1PARP3PIM1PIM2
Hydrochloric Acid SCHEMBL8799095 0.80 PARP1 (0.43) PARP1PARP3PIM1PIM2
SCHEMBL8800588 0.80 PARP1 (0.45) PARP1PIM1PIM2
SCHEMBL8800208 0.78 PARP1 (0.50) PARP1PARP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525584-B1 6-Oxo-azepinoindole derivatives, process and intermediates for their preparation and medicaments containing them SOLVAY PHARM GMBH (DE) 1997-12-10 EP disclosed
US-5272143-A 6-oxoazepinoindole compounds, and pharmaceutical compositions containing them KALI-CHEMIE PHARMA GMBH (DE) 1993-12-21 US disclosed
EP-0525584-A1 6-Oxo-azepinoindole derivatives, process and intermediates for their preparation and medicaments containing them Kali-Chemie Pharma GmbH (DE) 1993-02-03 EP disclosed