SCHEMBL8799951

SCHEMBL8799951

Cc1cccc(Nc2cc(N3CCC(C(=O)N4CCCC4)CC3)ncn2)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.46
EP300 Q09472 1/20 0.45
CREBBP Q92793 1/20 0.45
ALDH1A1 P00352 2/20 0.45
MAP4K4 O95819 1/20 0.45
CHRM4 P08173 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PDGFRB P09619 1/20 0.44
RAB9A P51151 2/20 0.44
KDM4E B2RXH2 2/20 0.44
USP2 O75604 1/20 0.44
LIMK2 P53671 1/20 0.44
EGFR P00533 1/20 0.43
HSD17B10 Q99714 1/20 0.43
KMT2A Q03164 1/20 0.43
PIK3CA P42336 1/20 0.43
PRKDC P78527 1/20 0.43
ACKR3 P25106 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27322788 0.91 KDM4E (0.56) SCN9AEP300CREBBPALDH1A1CHRM4
SCHEMBL8798398 0.88 SCN9A (0.48) SCN9AALDH1A1SMN1; SMN2PDGFRBKDM4E
SCHEMBL27335944 0.86 USP2 (0.50) SCN9AALDH1A1PDGFRBKDM4EUSP2
SCHEMBL8798331 0.86 PDGFRB (0.47) SCN9AALDH1A1SMN1; SMN2PDGFRBKDM4E
SCHEMBL8808651 0.84 EP300 (0.47) EP300CREBBPALDH1A1RAB9AKDM4E
SCHEMBL8808658 0.84 EP300 (0.47) EP300CREBBPALDH1A1RAB9AKDM4E
SCHEMBL27323457 0.80 EGFR (0.53) SCN9APDGFRBEGFRPIK3CAPRKDC
SCHEMBL8315857 0.77 EGFR (0.49) SCN9ASMN1; SMN2EGFRKMT2APIK3CA
SCHEMBL8805243 0.77 EGFR (0.55) SCN9AEGFR
SCHEMBL8318909 0.77 BRAF (0.53) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed