SCHEMBL8801280

SCHEMBL8801280

CC(=O)N1CCc2cc(SSc3cc4c(cc3CC(F)(F)F)N(C(C)=O)CC4)c(CC(F)(F)F)cc21

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 8/20 0.50
CYP11B2 P19099 6/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
RECQL P46063 1/20 0.39
CYP11B1 P15538 1/20 0.39
POLB P06746 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7083408 0.80 NOTUM (0.57) NOTUMCYP11B2KDM4EALDH1A1HPGD
SCHEMBL8785820 0.75 NOTUM (0.51) NOTUMCYP11B2KDM4EALDH1A1HPGD
SCHEMBL7086213 0.74 HTR2C (0.59) NOTUMCYP11B2KDM4EALDH1A1HPGD
SCHEMBL8530059 0.69 HTR2A (0.57) NOTUMCYP11B2KDM4EALDH1A1HPGD
SCHEMBL7373998 0.69 NOTUM (0.59) NOTUMCYP11B2KDM4EALDH1A1HPGD
SCHEMBL7479611 0.69 NOTUM (0.59) NOTUMCYP11B2KDM4EALDH1A1HPGD
SCHEMBL8526767 0.68 NOTUM (0.49) NOTUMCYP11B2KDM4EALDH1A1HPGD
SCHEMBL29803331 0.68 NOTUM (0.60) NOTUMCYP11B2KDM4EALDH1A1HPGD
SCHEMBL22462287 0.68 NOTUM (0.60) NOTUMCYP11B2KDM4EALDH1A1HPGD
SCHEMBL30038606 0.67 NOTUM (0.78) NOTUMALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0807104-A2 HETEROCYCLIC COMPOUNDS POSSESSING 5HT 2C? RECEPTOR ANTAGONIST ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1997-11-19 EP disclosed