SCHEMBL8801679

SCHEMBL8801679

NC[C@H]1CNC(=O)c2cccc3[nH]cc1c23

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.50
HTR6 P50406 1/20 0.35
HTR2A P28223 2/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
PARP3 Q9Y6F1 1/20 0.33
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8800208 1.00 PARP1 (0.50) PARP1HTR6HTR2AHTR2CHTR2B
SCHEMBL8799810 1.00 PARP1 (0.50) PARP1HTR6HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL8800428 0.99 PARP1 (0.49) PARP1HTR6HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL8801830 0.99 PARP1 (0.49) PARP1HTR6HTR2AHTR2CHTR2B
Water SCHEMBL8798203 0.99 PARP1 (0.49) PARP1HTR6HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL8800877 0.99 PARP1 (0.49) PARP1HTR6HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL8799094 0.97 PARP1 (0.48) PARP1HTR6HTR2AHTR2CHTR2B
Cadaverine Tartrate SCHEMBL8800774 0.90 PARP1 (0.41) PARP1HTR6PARP3ALDH1A1GAA
Cadaverine Tartrate SCHEMBL8801759 0.90 PARP1 (0.41) PARP1HTR6PARP3ALDH1A1GAA
SCHEMBL8798434 0.84 PARP1 (0.48) PARP1HTR2AHTR2CHTR2BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525584-B1 6-Oxo-azepinoindole derivatives, process and intermediates for their preparation and medicaments containing them SOLVAY PHARM GMBH (DE) 1997-12-10 EP disclosed
US-5272143-A 6-oxoazepinoindole compounds, and pharmaceutical compositions containing them KALI-CHEMIE PHARMA GMBH (DE) 1993-12-21 US disclosed