SCHEMBL880282

SCHEMBL880282

COc1ccccc1C1CC(=O)Nc2cc3c(cc21)OCCO3

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 10/20 1.00
LMNA P02545 8/20 1.00
ALDH1A1 P00352 1/20 1.00
HPGD P15428 1/20 1.00
TDP1 Q9NUW8 1/20 1.00
SMN1; SMN2 Q16637 9/20 0.78
TP53 P04637 7/20 0.78
NPSR1 Q6W5P4 4/20 0.78
MAPK1 P28482 3/20 0.78
ALOX15 P16050 2/20 0.78
GAA P10253 2/20 0.74
HSD17B10 Q99714 1/20 0.74
POLB P06746 1/20 0.71
MEN1 O00255 1/20 0.67
KMT2A Q03164 1/20 0.67
RAB9A P51151 1/20 0.65
THRB P10828 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10280607 0.93 TSHR (0.87) TSHRLMNAALDH1A1HPGDTDP1
SCHEMBL21643939 0.87 TSHR (1.00) TSHRLMNAALDH1A1HPGDTDP1
SCHEMBL12470138 0.86 TSHR (0.76) TSHRLMNAALDH1A1HPGDTDP1
SCHEMBL12698422 0.81 TSHR (0.69) TSHRLMNAALDH1A1HPGDTDP1
SCHEMBL880277 0.81 TSHR (0.69) TSHRLMNAALDH1A1HPGDTDP1
SCHEMBL12469684 0.81 SMN1; SMN2 (1.00) TSHRLMNAALDH1A1HPGDTDP1
SCHEMBL29433738 0.81 SMN1; SMN2 (1.00) TSHRLMNAALDH1A1HPGDTDP1
SCHEMBL12698265 0.81 SMN1; SMN2 (1.00) TSHRLMNAALDH1A1HPGDTDP1
SCHEMBL17226016 0.81 SMN1; SMN2 (1.00) TSHRLMNAALDH1A1HPGDTDP1
SCHEMBL29433753 0.81 SMN1; SMN2 (1.00) TSHRLMNAALDH1A1HPGDTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8440705-B2 2,3,4,7,8,9-hexahydro-1H-cyclopenta[h]quinolin-2-one or 2,3,4,6,7,8-hexahydro-1H-cyclopenta[g]quinolin-2-one; Alzheimer's disease WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2013-05-14 US disclosed
EP-2433634-A2 Compounds, compositions and methods of inhibiting a-synuclein toxicity The Whitehead Institute for Biomedical Research (US) 2012-03-28 EP disclosed