SCHEMBL8807151

SCHEMBL8807151

COc1cc2ncnc(Nc3ccc(OCc4ccccc4Br)c(OC)c3)c2cc1OC

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 14/20 0.69
ABCG2 Q9UNQ0 4/20 0.69
CLK1 P49759 1/20 0.69
LCK P06239 3/20 0.67
KDR P35968 6/20 0.64
JAK3 P52333 2/20 0.63
ABCB1 P08183 1/20 0.63
ERBB2 P04626 3/20 0.62
EPHB2 P29323 3/20 0.62
GAK O14976 2/20 0.62
KDM4E B2RXH2 1/20 0.62
MAPK13 O15264 1/20 0.62
ABL1 P00519 1/20 0.62
CYP1A2 P05177 1/20 0.62
CDK1 P06493 1/20 0.62
CYP3A4 P08684 1/20 0.62
FBP1 P09467 1/20 0.62
CYP2D6 P10635 1/20 0.62
MAPT P10636 1/20 0.62
CYP2C9 P11712 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8810211 0.94 EGFR (0.63) EGFRABCG2CLK1LCKKDR
Hydrochloric Acid SCHEMBL8808866 0.91 EGFR (0.65) EGFRABCG2CLK1LCKKDR
Hydrochloric Acid SCHEMBL8812282 0.91 EGFR (0.60) EGFRABCG2CLK1LCKKDR
Hydrochloric Acid SCHEMBL8816054 0.91 ABCG2 (0.71) EGFRABCG2CLK1LCKKDR
Hydrochloric Acid SCHEMBL8933913 0.88 EGFR (0.61) EGFRABCG2CLK1LCKKDR
Hydrochloric Acid SCHEMBL8812010 0.85 EGFR (0.67) EGFRABCG2CLK1LCKKDR
SCHEMBL1387156 0.84 EGFR (0.75) EGFRABCG2CLK1LCKKDR
Hydrochloric Acid SCHEMBL8811182 0.84 EGFR (0.76) EGFRABCG2CLK1LCKKDR
Hydrochloric Acid SCHEMBL8809182 0.83 EGFR (0.67) EGFRABCG2CLK1LCKKDR
SCHEMBL5570070 0.83 EGFR (0.85) EGFRABCG2CLK1LCKKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0782570-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1997-07-09 EP disclosed
WO-1996009294-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1996-03-28 WO disclosed