SCHEMBL8808199

SCHEMBL8808199

COc1cc2c(cc1OC)CN(CCCCc1ccc(NC(=O)c3cnc4cc(C)c(C)cc4n3)cc1)CC2

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 19/20 0.74
ABCB1 P08183 14/20 0.74
CYP1A2 P05177 1/20 0.57
CYP2C8 P10632 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
ABCC1 P33527 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8806668 0.91 ABCG2 (0.89) ABCG2ABCB1CYP1A2CYP2C8CYP2D6
SCHEMBL8809128 0.89 ABCG2 (0.91) ABCG2ABCB1CYP1A2CYP2C8CYP2D6
SCHEMBL8809428 0.84 ABCB1 (0.89) ABCG2ABCB1
SCHEMBL8808055 0.84 ABCB1 (0.59) ABCG2ABCB1
SCHEMBL8809233 0.82 ABCG2 (0.78) ABCG2ABCB1CYP1A2CYP2C8CYP2D6
SCHEMBL8806738 0.81 ABCB1 (0.90) ABCG2ABCB1CYP1A2CYP2C8CYP2D6
SCHEMBL8809248 0.81 ABCG2 (0.68) ABCG2ABCB1CYP1A2CYP2C8CYP2D6
SCHEMBL8805935 0.81 ABCB1 (0.73) ABCG2ABCB1CYP1A2CYP2C8CYP2D6
SCHEMBL8807296 0.81 ABCG2 (0.79) ABCG2ABCB1CYP1A2CYP2C8CYP2D6
SCHEMBL8807751 0.80 ABCG2 (0.91) ABCG2ABCB1CYP1A2CYP2C8CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5663179-A CAN SENSITIZE MULTIDRUG RESISTANT CANCER CELLS TO CHEMOTHERAPEUTIC AGENTS LABORATOIRES GLAXO SA (FR) 1997-09-02 US disclosed
EP-0649410-B1 ANILIDE DERIVATIVES GLAXO LAB SA (FR) 1997-05-02 EP disclosed