SCHEMBL8809912

SCHEMBL8809912

OCCC1CCN(c2ccc3c(c2)OCO3)C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.53
NOTUM Q6P988 1/20 0.42
CMA1 P23946 1/20 0.41
ALDH1A1 P00352 3/20 0.39
ACHE P22303 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
HTR1A P08908 1/20 0.38
ADRA2A P08913 1/20 0.38
DRD2 P14416 1/20 0.38
ADRA2C P18825 1/20 0.38
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
DRD3 P35462 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
HSD17B10 Q99714 2/20 0.38
HPGD P15428 2/20 0.38
USP2 O75604 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8808612 0.81 KDM4E (0.42) KDM4ECMA1ALDH1A1DRD2DRD3
SCHEMBL21136256 0.81 KDM4E (0.44) KDM4ENOTUMCMA1ALDH1A1HSD17B10
SCHEMBL2939131 0.76 BPTF (0.40) KDM4EALDH1A1ACHECYP3A4CYP2D6
SCHEMBL2940165 0.75 BPTF (0.39) KDM4EALDH1A1ACHECYP3A4CYP2D6
SCHEMBL2939391 0.74 MAPT (0.41) KDM4ENOTUMALDH1A1CYP3A4CYP2D6
SCHEMBL7408420 0.74 NOTUM (0.60) NOTUM
SCHEMBL14320304 0.74 MAPT (0.41) KDM4EALDH1A1ADRA2CHSD17B10USP2
SCHEMBL7801882 0.73 NOTUM (0.51) KDM4ENOTUMALDH1A1ACHEADRA1D
SCHEMBL6393391 0.72 CMA1 (0.49) KDM4ECMA1ALDH1A1HTR1AADRA2A
SCHEMBL2940577 0.71 NOTUM (0.44) NOTUMBPTFMAPTITGB2ICAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777666-A1 NOVEL SUBSTITUTED PIPERIDINES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES MERRELL PHARMACEUTICALS INC. (US) 1997-06-11 EP disclosed
WO-1996006094-A1 NOVEL SUBSTITUTED PIPERIDINES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES MERRELL PHARMACEUTICALS INC. (US) 1996-02-29 WO disclosed