SCHEMBL8812475

SCHEMBL8812475

CCc1oncc1C(=O)Nc1ccc(OC(F)(F)F)cc1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 5/20 0.75
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
THRB P10828 2/20 0.50
MAPT P10636 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
GMNN O75496 1/20 0.50
LMNA P02545 1/20 0.50
TP53 P04637 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
HTR1A P08908 1/20 0.50
PIM1 P11309 1/20 0.50
CYP2C9 P11712 1/20 0.50
MAOA P21397 1/20 0.50
SLC6A2 P23975 1/20 0.50
HTR2A P28223 1/20 0.50
AGTR1 P30556 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8808706 0.91 DHODH (0.62) DHODHMEN1KMT2ANPC1RAB9A
SCHEMBL8811917 0.85 DHODH (0.65) DHODHNPC1RAB9ATHRBMAPT
SCHEMBL11497402 0.84 DHODH (0.73) DHODHMEN1KMT2ANPC1RAB9A
SCHEMBL8811643 0.84 DHODH (0.73) DHODHMEN1KMT2ANPC1RAB9A
SCHEMBL8812402 0.82 DHODH (0.53) DHODHMEN1KMT2ANPC1RAB9A
SCHEMBL8810575 0.80 DHODH (0.51) DHODHNPC1RAB9ATHRBSMN1; SMN2
SCHEMBL8808868 0.80 DHODH (0.51) DHODHMEN1KMT2ANPC1RAB9A
SCHEMBL11493670 0.79 DHODH (0.66) DHODHNPC1RAB9ATHRBMAPT
Toluene SCHEMBL11494674 0.77 DHODH (0.64) DHODHNPC1RAB9ATHRBMAPT
SCHEMBL8809721 0.77 DHODH (0.48) DHODHMEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0527736-B1 ISOXAZOLE-4-CARBOXAMIDES AND HYDROXYALKYLIDENE-CYANOACETAMIDES, DRUGS CONTAINING THESE COMPOUNDS AND USE OF SUCH DRUGS HOECHST AG (DE) 1997-04-16 EP disclosed
US-5532259-A ANTITUMOR HOECHST AKTIENGESELLSCHAFT (DE) 1996-07-02 US disclosed
US-5494911-A TREATING LEUKEMIA, SARCOMA, CARCINOMA, LYMPHOMA, SKIN CANCER HOECHST AKTIENGESELLSCHAFT (DE) 1996-02-27 US disclosed
EP-0527736-A1 ISOXAZOLE-4-CARBOXAMIDES AND HYDROXYALKYLIDENE-CYANOACETAMIDES, DRUGS CONTAINING THESE COMPOUNDS AND USE OF SUCH DRUGS. HOECHST AG (DE) 1993-02-24 EP disclosed
WO-1991017748-A1 ISOXAZOLE-4-CARBOXAMIDES AND HYDROXYALKYLIDENE-CYANOACETAMIDES, DRUGS CONTAINING THESE COMPOUNDS AND USE OF SUCH DRUGS HOECHST AKTIENGESELLSCHAFT (DE) 1991-11-28 WO disclosed