SCHEMBL8814712

SCHEMBL8814712

COc1cccc2c1CCCC2CN(C)CCc1ccc2c(=O)ccoc2c1

nearest known ligand 0.78

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 4/20 0.78
HTR1A P08908 3/20 0.78
ADRA2A P08913 1/20 0.78
ADRA2B P18089 1/20 0.78
ADRA2C P18825 1/20 0.78
DRD4 P21917 1/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8814477 0.93 SLC6A4 (0.75) SLC6A4HTR1AADRA2AADRA2BADRA2C
SCHEMBL8814950 0.88 SLC6A4 (1.00) SLC6A4HTR1AADRA2AADRA2BADRA2C
SCHEMBL647243 0.88 SLC6A4 (1.00) SLC6A4HTR1AADRA2AADRA2BADRA2C
SCHEMBL9327727 0.87 SLC6A4 (0.66) SLC6A4HTR1AADRA2AADRA2BADRA2C
SCHEMBL9326564 0.87 SLC6A4 (0.68) SLC6A4HTR1AADRA2AADRA2BADRA2C
SCHEMBL9326970 0.86 SLC6A4 (0.75) SLC6A4HTR1AADRA2AADRA2BADRA2C
SCHEMBL8806272 0.86 SLC6A4 (0.86) SLC6A4HTR1AADRA2AADRA2BADRA2C
SCHEMBL9325372 0.84 SLC6A4 (0.89) SLC6A4HTR1AADRA2AADRA2BADRA2C
SCHEMBL9325382 0.84 SLC6A4 (0.89) SLC6A4HTR1AADRA2AADRA2BADRA2C
SCHEMBL8812074 0.84 SLC6A4 (0.72) SLC6A4HTR1AADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0646112-A4 TERTIARY AND SECONDARY AMINES AS ALPHA-2 ANTAGONISTS AND SEROTONIN UPTAKE INHIBITORS. ABBOTT LAB (US) 1997-04-02 EP disclosed
EP-0646112-A1 TERTIARY AND SECONDARY AMINES AS ALPHA-2 ANTAGONISTS AND SEROTONIN UPTAKE INHIBITORS ABBOTT LABORATORIES (US) 1995-04-05 EP disclosed
US-5288749-A Treating central nervous system or cardiovascular disorders ABBOTT LABORATORIES (US) 1994-02-22 US disclosed
WO-1993012754-A2 TERTIARY AND SECONDARY AMINES AS ALPHA-2 ANTAGONISTS AND SEROTONIN UPTAKE INHIBITORS ABBOTT LABORATORIES (US) 1993-07-08 WO disclosed