SCHEMBL8814751

SCHEMBL8814751

COc1cccc(-c2nc(-c3ccccn3)nc3ccccc23)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.64
ABCG2 Q9UNQ0 3/20 0.64
ADORA2A P29274 1/20 0.62
MAPT P10636 6/20 0.58
NPSR1 Q6W5P4 2/20 0.58
ALDH1A1 P00352 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
NPC1 O15118 1/20 0.58
PKM P14618 1/20 0.58
GRM5 P41594 1/20 0.58
RAB9A P51151 1/20 0.58
GAA P10253 1/20 0.58
CYP1A2 P05177 4/20 0.56
CYP3A4 P08684 4/20 0.56
CYP2C9 P11712 3/20 0.56
CYP2B6 P20813 2/20 0.56
AHR P35869 2/20 0.56
NR1I3 Q14994 2/20 0.56
VDR P11473 1/20 0.56
LMNA P02545 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23996434 0.87 METAP1 (0.59) ABCB1ABCG2MAPTNPSR1ALDH1A1
SCHEMBL24589752 0.86 METAP1 (0.57) ABCB1ABCG2MAPTNPSR1ALDH1A1
SCHEMBL8816575 0.85 ADORA2A (0.62) ABCB1ABCG2ADORA2AMAPTALDH1A1
SCHEMBL8819286 0.85 ADORA2A (0.62) ABCB1ABCG2ADORA2AMAPTALDH1A1
SCHEMBL8817283 0.84 ADORA2A (0.67) ABCB1ABCG2ADORA2AMAPTALDH1A1
SCHEMBL8815504 0.84 ADORA2A (0.60) ABCB1ABCG2ADORA2AMAPTALDH1A1
SCHEMBL6121390 0.83 ADORA2A (0.62) ABCB1ABCG2ADORA2AMAPTALDH1A1
SCHEMBL6120334 0.83 ADORA2A (0.62) ABCB1ABCG2ADORA2AMAPTALDH1A1
SCHEMBL8819077 0.83 ADORA2A (0.56) ABCB1ABCG2ADORA2AMAPTALDH1A1
SCHEMBL2913642 0.83 METAP1 (0.64) MAPTNPSR1ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012066122-A1 2 - (PYRIDIN- 2 -YL) -QUINAZOLINE DERIVATIVES AND THEIR USE AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-05-24 WO disclosed