SCHEMBL881500

SCHEMBL881500

Cc1nn(C)c(Oc2ccc(F)c(F)c2)c1C(=O)N[C@@H](C)c1ccc(C=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 6/20 0.56
CYP1A2 P05177 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP3A4 P08684 1/20 0.47
PTGER2 P43116 1/20 0.45
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
PHGDH O43175 6/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.38
ACACB O00763 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL881393 0.88 PTGER4 (0.72) PTGER4CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL15249968 0.86 PTGER4 (0.62) PTGER4CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL26416612 0.79 PTGER4 (0.68) PTGER4CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL26416727 0.79 PTGER4 (0.63) PTGER4CYP1A2CYP2C9CYP2C19PTGER2
SCHEMBL26416614 0.79 PTGER4 (0.57) PTGER4CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL24861754 0.77 PTGER4 (0.58) PTGER4PTGER2PHGDHACACB
SCHEMBL15250004 0.77 PTGER4 (0.60) PTGER4CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL881184 0.77 PTGER4 (0.70) PTGER4CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL15249899 0.76 PTGER4 (0.79) PTGER4PTGER2PHGDH
SCHEMBL24861773 0.76 PTGER4 (0.75) PTGER4PTGER2PHGDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012039972-A1 PHARMACEUTICAL COMPOSITION EISAI R&D MANAGEMENT CO., LTD. (JP) 2012-03-29 WO disclosed