SCHEMBL8817927

SCHEMBL8817927

O=c1cc(O)c2c(Cl)cccc2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.53
ALDH1A1 P00352 1/20 0.53
DAO P14920 2/20 0.51
GRIN2D O15399 2/20 0.51
GRIN3B O60391 2/20 0.51
GRIN1 Q05586 2/20 0.51
GRIN2A Q12879 2/20 0.51
GRIN2B Q13224 2/20 0.51
GRIN2C Q14957 2/20 0.51
GRIN3A Q8TCU5 2/20 0.51
ERCC5 P28715 1/20 0.50
FEN1 P39748 1/20 0.50
HTT P42858 2/20 0.45
PBRM1 Q86U86 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
DYRK1A Q13627 1/20 0.42
CCNB2 O95067 1/20 0.42
CDK1 P06493 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6579538 0.80 GRIN2D (0.53) KDM4EALDH1A1GRIN2DGRIN3BGRIN1
SCHEMBL27030273 0.79 KDM4E (0.53) KDM4EALDH1A1DAOFEN1HTT
SCHEMBL29830210 0.79 KDM4E (0.53) KDM4EALDH1A1DAOFEN1HTT
SCHEMBL17504437 0.78 ERCC5 (0.46) KDM4EALDH1A1DAOGRIN2DGRIN3B
SCHEMBL9393158 0.76 DAO (0.66) DAOGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL13730103 0.75 ABCG2 (0.53) KDM4EALDH1A1MEN1KMT2A
SCHEMBL2741026 0.74 PDPK1 (0.44) KDM4EALDH1A1DAOGRIN2DGRIN3B
SCHEMBL31619545 0.73 ERCC5 (0.53) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6009055 0.73 ERCC5 (0.53) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL12668292 0.73 ERN1 (0.57) KDM4EALDH1A1DAOERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0805809-A2 AZA AND AZA (N-OXY) ANALOGS OF GLYCINE/NMDA RECEPTOR ANTAGONISTS State of Oregon through Oregon State Board of Higher Education for and on behalf of Oregon Health Sc. Univ. & Univ. of Oregon (US) 1997-11-12 EP disclosed