SCHEMBL8819831

SCHEMBL8819831

O=C(O)CC1=CCC=CC=N1

nearest known ligand 0.31

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 2/20 0.31
GABRB2 P47870 2/20 0.31
HSD17B10 Q99714 1/20 0.31
AKR1B1 P15121 1/20 0.30
GABRP O00591 1/20 0.30
GABRD O14764 1/20 0.30
GABRA1 P14867 1/20 0.30
GABRB1 P18505 1/20 0.30
GABRG2 P18507 1/20 0.30
GABRB3 P28472 1/20 0.30
GABRA3 P34903 1/20 0.30
GABRA2 P47869 1/20 0.30
GABRA4 P48169 1/20 0.30
GABRE P78334 1/20 0.30
GABRA6 Q16445 1/20 0.30
GABRG1 Q8N1C3 1/20 0.30
GABRG3 Q99928 1/20 0.30
GABRQ Q9UN88 1/20 0.30
QPCT Q16769 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23829540 0.78
SCHEMBL18951794 0.74
SCHEMBL19265452 0.69
SCHEMBL6675097 0.65 AKR1B1 (0.30) AKR1B1
SCHEMBL25876502 0.65 AKR1B1 (0.30) AKR1B1
SCHEMBL599997 0.63
SCHEMBL10770752 0.63 AKR1B1 (0.31) GABRA5GABRB2AKR1B1GABRPGABRD
SCHEMBL2340346 0.61 AKR1B1 (0.33) AKR1B1
SCHEMBL18951801 0.59
SCHEMBL18951799 0.59

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997047624-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1997-12-18 WO disclosed
WO-1997047625-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1997-12-18 WO disclosed