SCHEMBL8823905

SCHEMBL8823905

COC(=O)c1ccc(C(=O)Cl)cc1.O=C(Cl)N1CCCc2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.56
ALDH1A1 P00352 3/20 0.56
NOTUM Q6P988 1/20 0.53
PDE4A P27815 1/20 0.53
PDE4B Q07343 1/20 0.53
PDE4C Q08493 1/20 0.53
PDE4D Q08499 1/20 0.53
SMN1; SMN2 Q16637 3/20 0.52
MAPT P10636 2/20 0.51
LMNA P02545 2/20 0.50
HPGD P15428 2/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
KDM4E B2RXH2 1/20 0.49
GAA P10253 1/20 0.49
PKM P14618 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
AVPR2 P30518 1/20 0.49
AVPR1A P37288 1/20 0.49
POLB P06746 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7345049 0.85 TSHR (0.76) TSHRALDH1A1PDE4APDE4BPDE4C
SCHEMBL30592391 0.83 SMN1; SMN2 (0.74) TSHRALDH1A1NOTUMSMN1; SMN2MAPT
SCHEMBL330273 0.83 SMN1; SMN2 (0.74) TSHRALDH1A1NOTUMSMN1; SMN2MAPT
SCHEMBL7349843 0.80 AVPR2 (0.72) TSHRALDH1A1LMNAHPGDKMT2A
SCHEMBL4863174 0.78 SMN1; SMN2 (0.67) TSHRALDH1A1NOTUMSMN1; SMN2MAPT
SCHEMBL4861742 0.77 MAPT (0.72) ALDH1A1SMN1; SMN2MAPTLMNAPKM
SCHEMBL23632960 0.77 MEN1 (0.53) TSHRALDH1A1NOTUMPDE4APDE4B
SCHEMBL30898774 0.77 MEN1 (0.53) TSHRALDH1A1NOTUMPDE4APDE4B
SCHEMBL7359695 0.77 AVPR1A (0.67) AVPR1A
SCHEMBL19260249 0.77 HDAC1 (0.72) ALDH1A1MAPTKDM4EGAATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997049668-A1 INHIBITIORS OF CYSTEINE PROTEASE SMITHKLINE BEECHAM CORPORATION (US) 1997-12-31 WO disclosed