SCHEMBL8826271

SCHEMBL8826271

C[C@@H](NCc1ccc(Oc2ccccc2)cc1)c1cccc2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 5/20 0.51
POLB P06746 1/20 0.48
ACP3 P15309 1/20 0.47
CARM1 Q86X55 1/20 0.46
PRMT6 Q96LA8 1/20 0.46
HRH3 Q9Y5N1 1/20 0.44
MAPK14 Q16539 1/20 0.44
HTT P42858 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MLNR O43193 1/20 0.43
ABCB11 O95342 1/20 0.43
ADRB1 P08588 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
CYP2D6 P10635 1/20 0.43
CHRM1 P11229 1/20 0.43
DRD2 P14416 1/20 0.43
ADRA2C P18825 1/20 0.43
CHRM3 P20309 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15131044 0.90 CASR (0.52) CASRPOLBACP3HTTKDM4E
SCHEMBL2341650 0.87 POLB (0.61) CASRPOLBACP3HTTMLNR
SCHEMBL15131229 0.87 POLB (0.61) CASRPOLBACP3HTTMLNR
SCHEMBL5193705 0.87 POLB (0.61) CASRPOLBACP3HTTMLNR
Hydrochloric Acid SCHEMBL31355096 0.86 CASR (0.60) CASRPOLBACP3HTTSMN1; SMN2
Hydrochloric Acid SCHEMBL3067899 0.86 CASR (0.60) CASRPOLBACP3HTTSMN1; SMN2
Hydrochloric Acid SCHEMBL3082165 0.86 CASR (0.60) CASRPOLBACP3HTTSMN1; SMN2
Hydrochloric Acid SCHEMBL607723 0.86 CASR (0.60) CASRPOLBACP3HTTSMN1; SMN2
SCHEMBL3348544 0.85 CASR (0.46) CASRCARM1PRMT6HRH3OPRM1
SCHEMBL2457278 0.85 CASR (0.46) CASRCARM1PRMT6HRH3OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5631401-A Inhibitors of protein farnesyltransferase and squalene synthase ABBOTT LABORATORIES (US) 1997-05-20 US disclosed
WO-1995021815-A1 CYCLOBUTANE DERIVATIVES AND THEIR USE AS INHIBITORS OF PROTEIN FARNESYLTRANSFERASE AND SQUALENE SYNTHASE ABBOTT LABORATORIES (US) 1995-08-17 WO disclosed