SCHEMBL8827697

SCHEMBL8827697

O=C(Nc1ccc(C(=O)N2CCCCc3cc(Cl)ccc32)cn1)c1ccccc1OCCO

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 4/20 0.50
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
AVPR1A P37288 2/20 0.46
IDO1 P14902 1/20 0.46
KCNH2 Q12809 1/20 0.46
F10 P00742 3/20 0.46
OXTR P30559 1/20 0.44
MAPT P10636 2/20 0.43
SLC12A2 P55011 1/20 0.43
WNK1 Q9H4A3 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8827696 0.95 AVPR2 (0.49) AVPR2HDAC1HDAC6AVPR1AIDO1
SCHEMBL8827668 0.93 AVPR2 (0.49) AVPR2HDAC1HDAC6AVPR1AIDO1
SCHEMBL8827612 0.91 AVPR2 (0.54) AVPR2HDAC1HDAC6AVPR1AIDO1
SCHEMBL8827569 0.90 AVPR2 (0.49) AVPR2HDAC1HDAC6AVPR1AIDO1
Hydrochloric Acid SCHEMBL8827701 0.90 F10 (0.51) AVPR2HDAC1HDAC6AVPR1AIDO1
SCHEMBL8827580 0.89 AVPR2 (0.46) AVPR2HDAC1HDAC6AVPR1AIDO1
SCHEMBL8827570 0.88 AVPR2 (0.49) AVPR2HDAC1HDAC6AVPR1AIDO1
SCHEMBL8827579 0.88 AVPR2 (0.52) AVPR2HDAC1HDAC6AVPR1AIDO1
SCHEMBL7354914 0.76 AVPR2 (0.53) AVPR2AVPR1A
Hydrochloric Acid SCHEMBL7351822 0.76 AVPR2 (0.52) AVPR2AVPR1AIDO1KCNH2OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5677299-A VASOPRESSIN OR OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1997-10-14 US disclosed
US-5498609-A Benzoazepinyl compounds as oxytocin and vasopressin antagonists OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1996-03-12 US disclosed
EP-0612319-A1 BENZOHETEROCYCLIC COMPOUNDS AS OXYTOCIN AND VASOPRESSIN ANTAGONISTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-08-31 EP disclosed
WO-1994004525-A1 BENZOHETEROCYCLIC COMPOUNDS AS OXYTOCIN AND VASOPRESSIN ANTAGONISTS OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1994-03-03 WO disclosed