SCHEMBL8835682

SCHEMBL8835682

NC(=O)C(Nn1cc(Cl)c2ccccc21)C(Nn1cc(Cl)c2ccccc21)C(N)=O

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 5/20 0.37
CNR2 P34972 2/20 0.37
KMT2A Q03164 3/20 0.36
ATM Q13315 1/20 0.36
MAPT P10636 4/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 3/20 0.34
EGFR P00533 1/20 0.34
SRC P12931 1/20 0.34
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33
NOTUM Q6P988 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
RECQL P46063 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9433290 0.76 KDM4E (0.41) KMT2AATMMAPTALDH1A1KDM4E
SCHEMBL8836337 0.74 KMT2A (0.38) KMT2AMAPTALDH1A1KDM4ENPC1
SCHEMBL8835680 0.73 KDM4E (0.36) KMT2AMAPTALDH1A1KDM4E
SCHEMBL9433286 0.73 KDM4E (0.36) KMT2AMAPTALDH1A1KDM4E
SCHEMBL8836625 0.69 SLC6A2 (0.44) CNR1CNR2KMT2AMAPTALDH1A1
SCHEMBL7238496 0.65 CYP1A2 (0.42) KMT2AATMMAPTALDH1A1KDM4E
SCHEMBL8836209 0.64 TSHR (0.40) CNR1CNR2KMT2AMAPTALDH1A1
SCHEMBL5693076 0.64 CA1 (0.43) KMT2A
SCHEMBL29037094 0.64 NOTUM (0.62) KMT2AATMMAPTALDH1A1KDM4E
SCHEMBL27774897 0.64 KMT2A (0.65) KMT2AMAPTALDH1A1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5646300-A NEUROPROTECTIVE AGENTS HOECHST MARION ROUSSEL, INC. (US) 1997-07-08 US disclosed
US-5591866-A NEUROPROTECTIVE AGENTS HOECHST MARION ROUSSEL INC. (US) 1997-01-07 US disclosed
US-5565579-A NEUROPROTECTIVE AGENT HOECHST MARION ROUSSEL INC. (US) 1996-10-15 US disclosed
EP-0563916-B1 (1H-Indol-1-yl)-2-(amino)acetamides and related (1H-indol-1-yl)-(aminoalkyl)amides, intermediates and a process for their preparation and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1995-08-16 EP disclosed
US-5319096-A Neuroprotective agent HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-06-07 US disclosed
EP-0563916-A1 (1H-Indol-1-yl)-2-(amino)acetamides and related (1H-indol-1-yl)-(aminoalkyl)amides, intermediates and a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-10-06 EP disclosed