SCHEMBL8846069

SCHEMBL8846069

[CH]=Cc1c(C(C)C)nc(C(C)C)c(COCc2ccccc2)c1-c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GCGR P47871 15/20 0.50
ESR1 P03372 1/20 0.46
HMGCR P04035 1/20 0.46
CHRM1 P11229 1/20 0.46
TBXA2R P21731 1/20 0.46
PDE4A P27815 1/20 0.46
ADRA1A P35348 1/20 0.46
AR P10275 3/20 0.43
DHODH Q02127 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6958682 0.89 AR (0.53) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL6963764 0.85 ESR1 (0.50) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL9261550 0.85 ESR1 (0.50) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL6958229 0.83 GCGR (0.70) GCGR
SCHEMBL9270541 0.78 HMGCR (0.62) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL9270549 0.78 HMGCR (0.62) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL6956310 0.77 HMGCR (0.60) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL9265076 0.76 GCGR (0.56) GCGRAR
SCHEMBL27299931 0.76 HMGCR (0.71) ESR1HMGCRCHRM1TBXA2RPDE4A
SCHEMBL6961134 0.76 HMGCR (0.64) HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641762-B1 Process for preparation of 5-hydroxy-3-ketoester derivative and optically active substance thereof UBE INDUSTRIES (JP) 1997-05-28 EP disclosed
US-5457225-A Process for preparation of 5-hydroxy-3-ketoester derivative and optically active substance thereof UBE INDUSTRIES LTD. (JP) 1995-10-10 US disclosed
EP-0641762-A1 Process for preparation of 5-hydroxy-3-ketoester derivative and optically active substance thereof UBE INDUSTRIES, LTD. (JP) 1995-03-08 EP disclosed