SCHEMBL8852147

SCHEMBL8852147

CN(Cc1ccccc1)c1ncnc2c(N3CCOCC3)nc(N3CCC(N)CC3)nc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.43
POLB P06746 1/20 0.41
ALDH1A1 P00352 4/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KDM4E B2RXH2 2/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
ADK P55263 1/20 0.40
PIK3CB P42338 1/20 0.39
PDE10A Q9Y233 2/20 0.38
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
KHK P50053 1/20 0.38
LMNA P02545 2/20 0.38
HTT P42858 1/20 0.38
NAPEPLD Q6IQ20 1/20 0.38
STK4 Q13043 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL9232767 0.96 TSHR (0.40) TSHRPOLBALDH1A1NPSR1KDM4E
SCHEMBL8851415 0.91 TSHR (0.43) TSHRPOLBALDH1A1NPSR1KDM4E
SCHEMBL9231518 0.89 TSHR (0.47) TSHRPOLBALDH1A1NPSR1KDM4E
SCHEMBL8851394 0.89 POLB (0.44) TSHRPOLBALDH1A1NPSR1KDM4E
SCHEMBL8851425 0.89 TSHR (0.41) TSHRPOLBALDH1A1NPSR1KDM4E
SCHEMBL8851055 0.89 HTT (0.42) TSHRPOLBALDH1A1NPSR1KDM4E
SCHEMBL8851867 0.89 TSHR (0.41) TSHRPOLBALDH1A1NPSR1KDM4E
SCHEMBL9233803 0.88 POLB (0.43) TSHRPOLBALDH1A1NPSR1KDM4E
SCHEMBL8851801 0.87 TSHR (0.45) TSHRPOLBALDH1A1NPSR1KDM4E
SCHEMBL10658223 0.87 KHK (0.44) TSHRPOLBALDH1A1NPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618814-A Trisubstituted pyrimido [5,4-d] pyrimidines for modulating multi-drug resistance and pharmaceutical compositions containing these compounds DR. KARL THOMAE GMBH (DE) 1997-04-08 US disclosed