SCHEMBL8855495

SCHEMBL8855495

CCCCCCOC(=O)n1c(C(F)(F)F)nc2c([N+](=O)[O-])cc(C(F)(F)F)cc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.42
CYP3A4 P08684 4/20 0.40
MAPK1 P28482 2/20 0.40
MAPT P10636 2/20 0.40
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40
TDP1 Q9NUW8 4/20 0.38
TSHR P16473 2/20 0.38
PLK1 P53350 1/20 0.35
HSP90AA1 P07900 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
ATF1 P18846 2/20 0.35
NFKB1 P19838 2/20 0.35
DCTPP1 Q9H773 1/20 0.34
PTPN1 P18031 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8855527 0.96 CYP3A4 (0.41) ESR1CYP3A4MAPK1MAPTLMNA
SCHEMBL8855582 0.92 ESR1 (0.39) ESR1CYP3A4MAPK1MAPTLMNA
SCHEMBL8855498 0.89 CYP3A4 (0.40) CYP3A4MAPK1MAPTLMNAGAA
SCHEMBL11643323 0.84 MAPT (0.39) CYP3A4MAPK1MAPTLMNAGAA
SCHEMBL11640778 0.84 PLK1 (0.38) CYP3A4MAPK1MAPTLMNAGAA
SCHEMBL8855574 0.84 CYP3A4 (0.42) CYP3A4MAPK1MAPTLMNAGAA
SCHEMBL8855585 0.82 TDP1 (0.44) CYP3A4MAPK1MAPTGAATDP1
SCHEMBL8855420 0.82 CYP3A4 (0.39) CYP3A4MAPK1MAPTLMNAGAA
SCHEMBL11639519 0.82 PLK1 (0.36) CYP3A4MAPK1MAPTLMNAGAA
SCHEMBL8855554 0.81 MAPK1 (0.37) CYP3A4MAPK1MAPTLMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5670485-A FEEDS FOR POULTRY WITH O-PHENYLENEDIAMINE OR BENZIMIDAZOLE WITH POLYETHER ANTIBIOTICS ELI LILLY AND COMPANY (US) 1997-09-23 US disclosed
US-4421759-A Methods for controlling fire ants ELI LILLY AND COMPANY (US) 1983-12-20 US disclosed
US-4122184-A Benzimidazole insecticides ELI LILLY AND COMPANY (US) 1978-10-24 US disclosed
US-3980784-A Control of animal parasites with benzimidazoles ELI LILLY AND COMPANY (US) 1976-09-14 US disclosed