SCHEMBL885929

SCHEMBL885929

CCN1C(=O)C(NC(=O)C2CC2)CCc2c1ccc(Nc1ncc(Cl)c(Nc3ccccc3S(=O)(=O)N(C)C)n1)c2OC

nearest known ligand 0.71

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 13/20 0.71
INSR P06213 10/20 0.71
KCNH2 Q12809 1/20 0.56
IGF1R P08069 1/20 0.47
EGFR P00533 1/20 0.45
EML4 Q9HC35 1/20 0.45
AXL P30530 5/20 0.44
ZAP70 P43403 2/20 0.44
PTK2 Q05397 2/20 0.44
AURKA O14965 1/20 0.44
AURKB Q96GD4 1/20 0.44
NEK2 P51955 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cyclopropane SCHEMBL16966197 0.93 ALK (0.73) ALKINSRKCNH2IGF1REGFR
SCHEMBL886496 0.92 ALK (0.70) ALKINSRKCNH2IGF1REGFR
SCHEMBL885875 0.92 ALK (0.70) ALKINSRKCNH2IGF1REGFR
SCHEMBL886701 0.91 ALK (0.70) ALKINSRKCNH2IGF1REGFR
SCHEMBL886323 0.88 ALK (0.78) ALKINSRKCNH2IGF1REGFR
SCHEMBL885835 0.88 ALK (0.78) ALKINSRKCNH2IGF1RAXL
SCHEMBL886199 0.83 ALK (1.00) ALKINSRKCNH2IGF1REGFR
SCHEMBL886105 0.83 ALK (0.57) ALKINSRKCNH2ZAP70PTK2
SCHEMBL886104 0.83 ALK (0.70) ALKINSR
SCHEMBL886360 0.79 ALK (0.78) ALKINSRKCNH2EGFRZAP70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8148391-B2 Fused bicyclic derivatives of 2,4-diaminopyrimidine as ALK and c-Met inhibitors CEPHALON, INC. (US) 2012-04-03 US disclosed