SCHEMBL8860744

SCHEMBL8860744

CCc1cc2c(-c3ccc[nH]c3=O)c(C(=O)N[S+]([O-])C3CC3)n(Cc3cc(C(N)=O)ccc3F)c2cc1F

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 1/20 0.40
KMT2A Q03164 1/20 0.33
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10255265 0.85 CYP2C8 (0.40) CYP2C8KMT2ACYP3A4CYP2C9CYP2C19
SCHEMBL862423 0.84 CYP2C8 (0.43) CYP2C8KMT2A
SCHEMBL832003 0.78 CYP2C8 (0.48) CYP2C8KMT2A
SCHEMBL831983 0.77 CYP2C8 (0.37) CYP2C8KMT2ACYP3A4CYP2C9CYP2C19
SCHEMBL862447 0.76 CYP2C8 (0.42) CYP2C8KMT2A
SCHEMBL831259 0.75 CYP2C8 (0.39) CYP2C8KMT2A
SCHEMBL831989 0.75 CYP2C8 (0.39) CYP2C8KMT2ACYP2C9
SCHEMBL831116 0.75 CYP2C8 (0.49) CYP2C8KMT2A
SCHEMBL862430 0.74 CYP2C8 (0.45) CYP2C8KMT2A
SCHEMBL862437 0.74 CYP2C8 (0.45) CYP2C8KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197842-B1 2, 3-SUBSTITUTED INDOLE DERIVATIVES FOR TREATING VIRAL INFECTIONS SCHERING CORP (US) 2012-05-23 EP disclosed