SCHEMBL8862016

SCHEMBL8862016

C#CCCCCCCCC(C)(C)[Si](O[Si](c1ccccc1)(c1ccccc1)C(C)(C)CCCCCCCC#C)(c1ccccc1)c1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.33
ALDH1A1 P00352 1/20 0.33
ALOX15 P16050 1/20 0.33
CYP1A2 P05177 2/20 0.31
CYP2D6 P10635 2/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
HSD17B10 Q99714 1/20 0.31
DRD2 P14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8862128 1.00 CYP3A4 (0.33) CYP3A4ALDH1A1ALOX15CYP1A2CYP2D6
SCHEMBL9311733 0.98 CYP3A4 (0.32) CYP3A4ALDH1A1ALOX15CYP1A2CYP2D6
SCHEMBL7036817 0.81 CYP3A4 (0.35) CYP3A4ALDH1A1ALOX15CYP1A2CYP2D6
SCHEMBL13192505 0.81 CYP3A4 (0.35) CYP3A4ALDH1A1ALOX15CYP1A2CYP2D6
SCHEMBL18215137 0.81 CYP3A4 (0.35) CYP3A4ALDH1A1ALOX15CYP1A2CYP2D6
SCHEMBL12048062 0.79 CYP3A4 (0.36) CYP3A4ALDH1A1ALOX15CYP1A2CYP2D6
SCHEMBL16878895 0.77 CYP3A4 (0.35) CYP3A4ALDH1A1ALOX15CYP1A2CYP2D6
SCHEMBL2481872 0.77 CYP3A4 (0.35) CYP3A4ALDH1A1ALOX15CYP1A2CYP2D6
SCHEMBL2480164 0.77 CYP3A4 (0.35) CYP3A4ALDH1A1ALOX15CYP1A2CYP2D6
SCHEMBL13295612 0.77 CYP3A4 (0.35) CYP3A4ALDH1A1ALOX15CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5656636-A TREATING PSORIASIS SMITHKLINE BEECHAM CORPORATION (US) 1997-08-12 US disclosed
US-5633258-A Pyridine compounds for treating leukotriene-related diseases SMITHKLINE BEECHAM CORPORATION (US) 1997-05-27 US disclosed
US-5631262-A Pyridine compounds for treating leukotriene-related diseases SMITHKLINE BEECHAM CORPORATION (US) 1997-05-20 US disclosed
WO-1994014797-A1 QUINOLINE COMPOUNDS AND THE TREATMENT OF LEUCOTRIENE RELATED DISEASES THEREWITH SMITHKLINE BEECHAM CORPORATION (US) 1994-07-07 WO disclosed