SCHEMBL8864802

SCHEMBL8864802

Cn1nc(-c2ccc(Cl)cc2)c2ccccc2c1=O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.67
NPSR1 Q6W5P4 3/20 0.64
GAA P10253 1/20 0.64
MAPT P10636 2/20 0.62
TP53 P04637 1/20 0.62
POLB P06746 1/20 0.62
TDP1 Q9NUW8 1/20 0.62
SMN1; SMN2 Q16637 4/20 0.62
ALDH1A1 P00352 2/20 0.62
PPARG P37231 1/20 0.59
NR2E3 Q9Y5X4 1/20 0.59
NCOR2 Q9Y618 1/20 0.59
ENPP1 P22413 2/20 0.58
HTT P42858 3/20 0.57
LMNA P02545 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8224982 0.86 HPGD (0.74) HPGDNPSR1MAPTTP53POLB
SCHEMBL8864677 0.85 HPGD (0.70) HPGDNPSR1GAAMAPTPOLB
SCHEMBL8864712 0.84 HPGD (0.63) HPGDNPSR1MAPTTP53POLB
SCHEMBL1376771 0.84 HPGD (0.71) HPGDNPSR1MAPTTP53POLB
SCHEMBL29382447 0.84 SMN1; SMN2 (0.70) HPGDNPSR1MAPTTP53POLB
SCHEMBL8864626 0.84 HPGD (0.67) HPGDNPSR1MAPTTP53POLB
SCHEMBL8865071 0.84 HPGD (0.67) HPGDNPSR1MAPTTP53POLB
SCHEMBL8864710 0.83 HPGD (0.60) HPGDNPSR1GAAMAPTPOLB
SCHEMBL8268002 0.82 HPGD (0.64) HPGDNPSR1GAAMAPTTP53
SCHEMBL8864836 0.81 HPGD (0.63) HPGDNPSR1MAPTTP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624922-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1997-04-29 US disclosed
EP-0597540-B1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC (US) 1996-06-05 EP disclosed
US-5380721-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1995-01-10 US disclosed
EP-0597540-A1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1994-05-18 EP disclosed