SCHEMBL8870519

SCHEMBL8870519

CC(C)(N)CCNCc1cccnc1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.61
CYP2D6 P10635 1/20 0.61
CHRM2 P08172 1/20 0.59
ALDH1A1 P00352 4/20 0.54
NPSR1 Q6W5P4 1/20 0.54
HTT P42858 2/20 0.50
LMNA P02545 1/20 0.50
SCN8A Q9UQD0 1/20 0.50
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
TP53 P04637 1/20 0.48
POLB P06746 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
RECQL P46063 1/20 0.46
NOS1 P29475 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17282183 0.87 CYP1A2 (0.65) CYP1A2CYP2D6CHRM2ALDH1A1NPSR1
SCHEMBL7992321 0.84 CYP1A2 (0.65) CYP1A2CYP2D6CHRM2ALDH1A1NPSR1
SCHEMBL19031318 0.81 CYP1A2 (0.83) CYP1A2CYP2D6CHRM2ALDH1A1NPSR1
SCHEMBL29875178 0.81 CYP1A2 (0.83) CYP1A2CYP2D6CHRM2ALDH1A1NPSR1
SCHEMBL5367032 0.81 CYP1A2 (0.65) CYP1A2CYP2D6CHRM2ALDH1A1NPSR1
SCHEMBL3405350 0.78 CHRM2 (0.74) CYP1A2CYP2D6CHRM2ALDH1A1NPSR1
SCHEMBL3738479 0.78 CYP1A2 (0.71) CYP1A2CYP2D6CHRM2ALDH1A1NPSR1
SCHEMBL11594897 0.78 CHRM2 (0.93) CYP1A2CYP2D6CHRM2ALDH1A1NPSR1
SCHEMBL13493227 0.77 CHRM2 (0.44) CYP1A2CYP2D6CHRM2LMNAHTR2A
SCHEMBL2861457 0.77 CYP1A2 (1.00) CYP1A2CYP2D6CHRM2ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5654323-A 2-NITROGEN-CONTAINING FUNCTIONAL GROUP-HALOBENZOTHIAZOLES; ANALGESICS; ANTIINFLAMMATORY AND HYPOTENSIVE AGENTS; INHIBITORS OF CYTOKINES (INCLUDING TUMOR NECROSIS FACTOR) AND PHOSPHOLIPASE; SEPTIC SHOCK ADIR ET COMPAGNIE (FR) 1997-08-05 US disclosed
US-5597819-A ANTIINFLAMMATORY AGENTS ADIR ET COMPAGNIE (FR) 1997-01-28 US disclosed
US-5550143-A Heterocyclic compounds ADIR ET COMPAGNIE (FR) 1996-08-27 US disclosed