SCHEMBL8874008

SCHEMBL8874008

COC(=O)c1cc(OC)c2c(=O)[nH]c(C)nc2c1OC

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.43
POLB P06746 2/20 0.43
GPR183 P32249 1/20 0.41
ALDH1A1 P00352 4/20 0.41
HPGD P15428 2/20 0.41
USP2 O75604 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MAPT P10636 2/20 0.38
NPSR1 Q6W5P4 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP3A4 P08684 1/20 0.37
KLK7 P49862 1/20 0.36
GAA P10253 1/20 0.36
TYMS P04818 1/20 0.36
BACE1 P56817 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4261933 0.74 PDE4A (0.44) KDM4EPOLBALDH1A1HPGDMAPT
SCHEMBL13255445 0.71 PARP1 (0.46) KDM4EALDH1A1HPGDMAPTNPSR1
SCHEMBL8874761 0.70 SMN1; SMN2 (0.52) KDM4EPOLBALDH1A1MAPTKMT2A
SCHEMBL25647629 0.69 PARP1 (0.49) KDM4EHSD17B10TYMS
SCHEMBL12237369 0.69 PDE4A (0.61) KDM4EALDH1A1HSD17B10MAPTGAA
SCHEMBL1553062 0.69 PDE4A (0.52) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL18643546 0.68 TYMS (0.43) KDM4EALDH1A1HPGDHSD17B10TYMS
SCHEMBL527419 0.68 PARP1 (0.60) KDM4EALDH1A1HPGDNPSR1KMT2A
SCHEMBL18643549 0.65 PDE3B (0.64) KDM4EHSD17B10TYMS
SCHEMBL25414495 0.65 PARP1 (0.48) KDM4EGPR183ALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639881-A ANTITUMOR AGENTS, TREATMENT OF BREAST CANCER ARIZONA BOARD OF REGENTS ACTING ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 1997-06-17 US disclosed