SCHEMBL8874666

SCHEMBL8874666

CCOC(=O)[C@H](CCc1ccccc1)N[C@H]1COc2ccccc2N(Cc2ccc(C(C)C)cc2)C1=O

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACE P12821 5/20 0.53
ABCB11 O95342 1/20 0.53
AGTR2 P50052 1/20 0.53
PDE3A Q14432 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
XIAP P98170 8/20 0.53
KDM4E B2RXH2 1/20 0.53
CYP3A4 P08684 1/20 0.53
NPY1R P25929 1/20 0.47
MME P08473 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8874659 1.00 ACE (0.53) ACEABCB11AGTR2PDE3ATDP1
SCHEMBL8873232 0.93 ACE (0.56) ACEABCB11AGTR2PDE3ATDP1
SCHEMBL8873239 0.93 ACE (0.56) ACEABCB11AGTR2PDE3ATDP1
SCHEMBL8873842 0.92 XIAP (0.53) ACEABCB11AGTR2PDE3ATDP1
SCHEMBL8873838 0.92 XIAP (0.53) ACEABCB11AGTR2PDE3ATDP1
SCHEMBL8874308 0.92 XIAP (0.56) ACEXIAPNPY1R
SCHEMBL8873349 0.92 XIAP (0.56) ACEXIAPNPY1R
SCHEMBL8874316 0.92 XIAP (0.56) ACEXIAPNPY1R
SCHEMBL8873347 0.92 XIAP (0.56) ACEXIAPNPY1R
SCHEMBL8875377 0.90 XIAP (0.54) ACEXIAPNPY1RMME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5610153-A ENZYME INHIBITORS; TREATMENT OF VASCULAR PROLIFERATION DISORDERS, STERILITY DYSFUNCTION, DYSMENORRHEA CIBA-GEIGY CORPORATION (US) 1997-03-11 US disclosed
EP-0673371-A1 BENZAZEPINONE DERIVATIVES Novartis AG (CH) 1995-09-27 EP disclosed
WO-1994013651-A1 BENZAZEPINONE DERIVATIVES CIBA-GEIGY AG (CH) 1994-06-23 WO disclosed