SCHEMBL8878445

SCHEMBL8878445

CNC(C)(C)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.52
SSTR4 P31391 2/20 0.45
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
CASR P41180 1/20 0.40
AHR P35869 1/20 0.37
TP53 P04637 1/20 0.37
KCNH2 Q12809 5/20 0.36
TMEM97 Q5BJF2 2/20 0.36
KIF11 P52732 2/20 0.35
SLC6A4 P31645 4/20 0.35
HTR2A P28223 3/20 0.35
CYP3A4 P08684 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A3 Q01959 1/20 0.34
CYP19A1 P11511 1/20 0.34
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL799541 0.77 TSHR (0.61) TSHRSSTR4HDAC3HDAC1HDAC2
SCHEMBL8804344 0.75 TSHR (0.48) TSHRSSTR4HDAC3HDAC1HDAC2
SCHEMBL9222314 0.75 HDAC3 (0.46) TSHRSSTR4HDAC3HDAC1HDAC2
SCHEMBL10347814 0.75 TSHR (0.58) TSHRSSTR4HDAC3HDAC1HDAC2
SCHEMBL11665761 0.75 TSHR (0.65) TSHRSSTR4HDAC3HDAC1HDAC2
SCHEMBL5301475 0.75 MEN1 (0.52) TSHRSLC6A4HTR2ASLC6A2SLC6A3
SCHEMBL10192309 0.73 TSHR (0.56) TSHRSSTR4HDAC3HDAC1HDAC2
SCHEMBL8192026 0.73 TSHR (0.56) TSHRSSTR4HDAC3HDAC1HDAC2
SCHEMBL2796185 0.73 TSHR (0.56) TSHRSSTR4HDAC3HDAC1HDAC2
SCHEMBL3075392 0.73 TSHR (0.56) TSHRSSTR4HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5621010-A ANTIHYPERCHOLESTEROLEMIA AND ANTIATHEROSCLEROSIS NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-04-15 US disclosed
EP-0625507-A2 Urea derivatives and their use as acat inhibitors NISSHIN FLOUR MILLING CO., LTD. (JP) 1994-11-23 EP disclosed