SCHEMBL8884152

SCHEMBL8884152

COC(=O)c1ccccc1N(CC(F)(F)F)C(=O)CBr

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.45
PDK2 Q15119 1/20 0.40
LMNA P02545 2/20 0.40
TSHR P16473 1/20 0.40
ALDH1A1 P00352 3/20 0.39
HSD17B10 Q99714 2/20 0.39
CFTR P13569 1/20 0.39
TSPO P30536 2/20 0.38
KDM4E B2RXH2 3/20 0.38
POLB P06746 2/20 0.38
ATM Q13315 1/20 0.38
SLC6A3 Q01959 2/20 0.37
GLA P06280 1/20 0.37
SLC6A4 P31645 1/20 0.37
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA5A P35218 1/20 0.35
CA9 Q16790 1/20 0.35
MAPT P10636 1/20 0.35
ALOX15 P16050 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8824661 0.81 KMT2A (0.47) KMT2ALMNATSHRALDH1A1HSD17B10
SCHEMBL7819216 0.77 KMT2A (0.55) KMT2ALMNATSHRALDH1A1HSD17B10
SCHEMBL9369081 0.76 KMT2A (0.54) KMT2ALMNATSHRALDH1A1HSD17B10
SCHEMBL26623920 0.72 KMT2A (0.55) KMT2APDK2LMNATSHRALDH1A1
SCHEMBL26627265 0.71 KMT2A (0.54) KMT2APDK2LMNATSHRALDH1A1
SCHEMBL12474134 0.70 KMT2A (0.53) KMT2ALMNATSHRALDH1A1HSD17B10
SCHEMBL28525712 0.70 KMT2A (0.53) KMT2ALMNATSHRALDH1A1HSD17B10
SCHEMBL30492227 0.69 KMT2A (0.64) KMT2ALMNATSHRALDH1A1HSD17B10
SCHEMBL13066502 0.69 KMT2A (0.64) KMT2ALMNATSHRALDH1A1HSD17B10
SCHEMBL4444645 0.68 KMT2A (0.67) KMT2ALMNATSHRALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658933-A Substituted heterocyclic carboxamide esters, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-08-19 US disclosed
US-5618812-A GASTRIN ANTAGONISTS; GASTROINTESTINAL DISORDERS MERCK SHARP & DOHME, LTD. (GB) 1997-04-08 US disclosed