SCHEMBL8891065

SCHEMBL8891065

CNC(=O)c1ccccc1C[C@H]1CC[C@H](Nc2nc(Nc3ccc(Cl)cc3)c3ccccc3n2)CC1

nearest known ligand 0.68

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 11/20 0.68
CTNNB1 P35222 4/20 0.46
TCF7L2 Q9NQB0 4/20 0.46
MERTK Q12866 2/20 0.44
CDK7 P50613 1/20 0.43
CDK9 P50750 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
APP P05067 1/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8891045 1.00 NPY5R (0.68) NPY5RCTNNB1TCF7L2MERTKCDK7
SCHEMBL8891241 0.90 NPY5R (0.68) NPY5RCTNNB1TCF7L2MERTKAPP
SCHEMBL8891254 0.90 NPY5R (0.68) NPY5RCTNNB1TCF7L2MERTKAPP
SCHEMBL8892092 0.84 NPY5R (0.62) NPY5RMERTKAPPBCHEACHE
SCHEMBL8892104 0.84 NPY5R (0.62) NPY5RMERTKAPPBCHEACHE
SCHEMBL8890729 0.83 NPY5R (0.72) NPY5RCTNNB1TCF7L2MERTKAPP
SCHEMBL8890766 0.83 NPY5R (0.72) NPY5RCTNNB1TCF7L2MERTKAPP
SCHEMBL8891621 0.81 NPY5R (1.00) NPY5RCTNNB1TCF7L2MERTKAPP
SCHEMBL8891244 0.80 NPY5R (1.00) NPY5RCTNNB1TCF7L2MERTKAPP
SCHEMBL8892081 0.80 NPY5R (0.76) NPY5RCTNNB1TCF7L2MERTKCDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020823-A2 2-AMINO QUINAZOLINE DERIVATIVES AS NPY RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 1997-06-12 WO claimed