SCHEMBL8891464

SCHEMBL8891464

COc1cccc(Nc2nc(Nc3ccc(CN)cc3)nc3ccccc23)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 4/20 0.69
KDM4E B2RXH2 2/20 0.64
HTT P42858 2/20 0.64
TAAR1 Q96RJ0 1/20 0.64
ABCG2 Q9UNQ0 7/20 0.60
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
ABCB1 P08183 5/20 0.59
PDE5A O76074 1/20 0.59
SLC2A1 P11166 1/20 0.58
MERTK Q12866 2/20 0.58
PAK4 O96013 1/20 0.56
PAK1 Q13153 1/20 0.56
ALDH1A1 P00352 1/20 0.55
MAPT P10636 1/20 0.55
HPGD P15428 1/20 0.55
ALOX12 P18054 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
RXFP1 Q9HBX9 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8890929 0.99 NPY5R (0.67) NPY5RKDM4EHTTTAAR1ABCG2
SCHEMBL8889343 0.91 NPY5R (0.79) NPY5RABCG2MEN1KMT2ASLC2A1
SCHEMBL8891851 0.91 NPY5R (0.78) NPY5RKDM4EHTTTAAR1ABCG2
Hydrochloric Acid SCHEMBL8890985 0.90 NPY5R (0.77) NPY5RHTTTAAR1ABCG2MEN1
Hydrochloric Acid SCHEMBL8899399 0.90 NPY5R (0.76) NPY5RKDM4EHTTTAAR1ABCG2
SCHEMBL8889167 0.90 NPY5R (0.76) NPY5RKDM4EHTTTAAR1ABCG2
Hydrochloric Acid SCHEMBL8907334 0.89 NPY5R (0.83) NPY5RKDM4EHTTTAAR1ABCG2
Hydrochloric Acid SCHEMBL8907425 0.89 HTT (0.75) NPY5RKDM4EHTTTAAR1ABCG2
SCHEMBL8889361 0.89 KDM4E (0.70) NPY5RKDM4EHTTTAAR1ABCG2
SCHEMBL8891586 0.89 NPY5R (0.65) NPY5RKDM4EHTTTAAR1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO claimed
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO disclosed