SCHEMBL8891659

SCHEMBL8891659

COC(=O)CCC[C@@H](OC(C)=O)c1cccc(Br)n1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.36
CNR2 P34972 2/20 0.34
CNR1 P21554 1/20 0.34
ALDH1A1 P00352 3/20 0.34
ALOX5 P09917 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
TSHR P16473 1/20 0.33
PPARG P37231 2/20 0.33
MAPT P10636 2/20 0.33
PPARA Q07869 1/20 0.33
LTB4R Q15722 1/20 0.32
HPGD P15428 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8893092 1.00 IRAK4 (0.36) IRAK4CNR2CNR1ALDH1A1ALOX5
SCHEMBL4839728 0.85 IRAK4 (0.36) IRAK4ALDH1A1ALOX5PPARG
SCHEMBL4839737 0.85 IRAK4 (0.36) IRAK4ALDH1A1ALOX5PPARG
SCHEMBL8892818 0.83 IRAK4 (0.42) IRAK4CNR2CNR1ALDH1A1NFKB1
SCHEMBL8891780 0.83 IRAK4 (0.42) IRAK4CNR2CNR1ALDH1A1NFKB1
SCHEMBL17441067 0.78 IRAK4 (0.36) IRAK4ALDH1A1ALOX5TSHRHPGD
SCHEMBL17440806 0.73 IRAK4 (0.38) IRAK4ALDH1A1
SCHEMBL24012874 0.72 IRAK4 (0.39) IRAK4ALDH1A1TSHRMAPTHPGD
SCHEMBL24012872 0.72 IRAK4 (0.39) IRAK4ALDH1A1TSHRMAPTHPGD
SCHEMBL9146179 0.72 HPGD (0.45) CNR2CNR1ALDH1A1TSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997037976-A1 NEW LEUKOTRIENE-B4 DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR USE AS MEDICAMENTS SCHERING AKTIENGESELLSHAFT (DE) 1997-10-16 WO disclosed