SCHEMBL8895819

SCHEMBL8895819

O=[N+]([O-])c1nccn1C[C@@H](O)CN1CC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.67
LMNA P02545 3/20 0.45
THRB P10828 1/20 0.45
CYP2C19 P33261 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
CA12 O43570 5/20 0.43
CA1 P00915 5/20 0.43
CA2 P00918 5/20 0.43
CA9 Q16790 5/20 0.43
TYMP P19971 3/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
OPRK1 P41145 1/20 0.41
TDP1 Q9NUW8 1/20 0.39
MAPT P10636 4/20 0.37
ALDH1A1 P00352 3/20 0.37
HTT P42858 2/20 0.37
RAD52 P43351 1/20 0.35
NPY1R P25929 1/20 0.34
NPY2R P49146 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8855534 1.00 KMT2A (0.67) KMT2ALMNATHRBCYP2C19L3MBTL1
SCHEMBL367134 1.00 KMT2A (0.67) KMT2ALMNATHRBCYP2C19L3MBTL1
SCHEMBL11352268 0.94 KMT2A (0.64) KMT2ALMNATHRBCYP2C19L3MBTL1
SCHEMBL11379553 0.94 KMT2A (0.64) KMT2ALMNATHRBCYP2C19L3MBTL1
Hydrochloric Acid SCHEMBL11376105 0.93 KMT2A (0.63) KMT2ALMNATHRBCYP2C19L3MBTL1
Pimonidazole SCHEMBL51977 0.93 KMT2A (0.63) KMT2ALMNATHRBCYP2C19L3MBTL1
Hydrochloric Acid SCHEMBL11379185 0.92 KMT2A (0.62) KMT2ALMNATHRBCYP2C19L3MBTL1
Pimonidazole SCHEMBL11390660 0.92 KMT2A (0.62) KMT2ALMNATHRBCYP2C19L3MBTL1
SCHEMBL12396375 0.91 KMT2A (0.78) KMT2ALMNATHRBCYP2C19CA12
SCHEMBL11350180 0.91 KMT2A (0.60) KMT2ALMNATHRBCYP2C19L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5659048-A CHEMOSENSITIZER, RADIOSENSITIZER ADMINISTERING TO PATIENTS WHOM ARE SENSITIVE TO RADIATION OR CHEMOTHERAPY BRITISH TECHNOLOGY GROUP LIMITED (GB) 1997-08-19 US disclosed
US-5543527-A ANTITUMOR AGENTS BRITISH TECHNOLOYG GROUP LIMITED (GB) 1996-08-06 US disclosed
US-5481000-A RADIOSENSITIZERS OR CHEMOSENSITIZERS; PATENT CLAIMS CHIRAL 3-/2-HYDROXY-3-/2-NITROIMIDAZOL-1-YL/PROPYL/-2-OXAZOLIDINONE, HAVING /S/ CONFIGURATION AT OH CARBON AND FREE OF /R/ CONFIGURATION WARNER-LAMBERT COMPANY (US) 1996-01-02 US disclosed
EP-0652870-A1 Process for preparing chiral (((2-bromoethyl)amino)methyl)-2-nitro-1H-imidazol-1- ethanol and related compounds WARNER-LAMBERT COMPANY (US) 1995-05-17 EP disclosed
US-5342959-A Process for preparing chiral [[(2-bromoethyl)-amino]methyl]-2-nitro-1H-imidazol-1-ethanol and related compounds WARNER-LAMBERT COMPANY (US) 1994-08-30 US disclosed
WO-1994015922-A1 NOVEL PROCESS FOR PREPARING CHIRAL [[(2-BROMOETHYL)AMINO]METHYL]-2-NITRO-1H-IMIDAZOL-1-ETHANOL AND RELATED COMPOUNDS WARNER LAMBERT COMPANY (US) 1994-07-21 WO disclosed