SCHEMBL8897218

SCHEMBL8897218

Cc1ccc(N2CN(CC(=O)O)C(=O)C23CCN(C(=O)OC(C)(C)C)CC3)cc1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NPC1L1 Q9UHC9 13/20 0.60
BDKRB2 P30411 2/20 0.58
OPRM1 P35372 1/20 0.50
OPRK1 P41145 1/20 0.50
DDR1 Q08345 3/20 0.47
GPR119 Q8TDV5 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1855447 0.92 NPC1L1 (0.70) NPC1L1BDKRB2OPRM1OPRK1DDR1
SCHEMBL8894157 0.90 NPC1L1 (0.59) NPC1L1BDKRB2OPRM1OPRK1DDR1
SCHEMBL17140929 0.83 NPC1L1 (0.65) NPC1L1BDKRB2OPRM1OPRK1DDR1
SCHEMBL8892630 0.83 NPC1L1 (0.67) NPC1L1BDKRB2OPRM1OPRK1DDR1
SCHEMBL20187144 0.82 NPC1L1 (0.66) NPC1L1OPRM1OPRK1DDR1
SCHEMBL20187070 0.82 NPC1L1 (0.66) NPC1L1BDKRB2DDR1
SCHEMBL8893884 0.81 NPC1L1 (0.56) NPC1L1BDKRB2OPRM1OPRK1DDR1
SCHEMBL20187219 0.81 NPC1L1 (0.74) NPC1L1DDR1
SCHEMBL20187150 0.81 NPC1L1 (0.64) NPC1L1DDR1
SCHEMBL5563023 0.80 NPC1L1 (0.64) NPC1L1BDKRB2OPRM1OPRK1DDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5610142-A Bradykinin antagonist pseudopeptide derivatives of substituted 4-keto-1,3,8-triazaspiro[4.5]decan-3-alkanoic acids SCIOS INC. (US) 1997-03-11 US disclosed