SCHEMBL8900482

SCHEMBL8900482

Cc1cccc(CN(C)CCN)c1

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CARM1 Q86X55 3/20 0.65
PRMT6 Q96LA8 1/20 0.65
PRMT8 Q9NR22 1/20 0.65
TAAR1 Q96RJ0 3/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
RECQL P46063 1/20 0.56
PRMT1 Q99873 3/20 0.52
IDO1 P14902 2/20 0.46
ACHE P22303 1/20 0.43
AOC3 Q16853 1/20 0.40
SIGMAR1 Q99720 2/20 0.40
HSP90AA1 P07900 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9903565 0.84 TAAR1 (0.58) CARM1PRMT6PRMT8TAAR1CYP2D6
SCHEMBL18138028 0.84 CYP2D6 (0.57) CARM1PRMT6PRMT8TAAR1CYP2D6
SCHEMBL18378603 0.84 CYP2D6 (0.57) CARM1PRMT6PRMT8TAAR1CYP2D6
SCHEMBL13175212 0.82 CYP2D6 (0.56) CARM1PRMT6PRMT8TAAR1CYP2D6
SCHEMBL21902241 0.81 CARM1 (0.62) CARM1PRMT6PRMT8TAAR1RECQL
SCHEMBL19049389 0.81 CARM1 (0.62) CARM1PRMT6PRMT8TAAR1PRMT1
SCHEMBL14174779 0.81 CYP2D6 (0.55) CARM1PRMT6PRMT8TAAR1CYP2D6
SCHEMBL12124993 0.79 CYP2D6 (0.53) TAAR1CYP2D6CYP2C9CYP2C19RECQL
SCHEMBL14492296 0.79 CYP2D6 (0.54) CARM1PRMT6TAAR1CYP2D6CYP2C9
SCHEMBL14174811 0.79 CYP2D6 (0.54) TAAR1CYP2D6CYP2C9CYP2C19RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-9100276-A None JP disclosed
EP-3498708-B1 DEUTERATED 3-(4,5-SUBSTITUTED PYRIMIDINAMINE) PHENYL DERIVATIVES AND APPLICATIONS THEREOF NANJING CHUANGTE PHARMACEUTICAL TECH CO LTD (CN) 2021-01-13 EP disclosed
EP-3747887-A1 CRYSTAL FORM OF MONOMETHANESULFONATE OF DEUTERATED 3-(4,5-SUBSTITUTED AMINOPYRIMIDINE)PHENYL COMPOUND, AND PREPARATION METHOD THEREFOR Nanjing Chuangte Pharmaceutical Technology Co., Ltd (CN) 2020-12-09 EP disclosed
EP-3498708-A1 DEUTERATED 3-(4,5-SUBSTITUTED PYRIMIDINAMINE) PHENYL DERIVATIVES AND APPLICATIONS THEREOF Nanjing Chuangte Pharmaceutical Technology Co., Ltd (CN) 2019-06-19 EP disclosed
JP-H09100276-A (R)-1-ETHYL-4-METHYLHEXAHYDRO-1H-1,4-DIAZEPINE DERIVATIVE AND MEDICINE CONTAINING THE SAME DAINIPPON PHARMACEUT CO LTD 1997-04-15 JP disclosed