SCHEMBL8900769

SCHEMBL8900769

COc1ccc2nc(Nc3ccc(OCc4ccccc4)cc3)nc(Nc3ccccc3)c2c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.72
ERBB2 P04626 6/20 0.72
NPY5R Q15761 1/20 0.63
SLC2A1 P11166 1/20 0.56
MERTK Q12866 4/20 0.53
ERBB4 Q15303 2/20 0.52
CHEK2 O96017 1/20 0.52
ROS1 P08922 1/20 0.52
FLT3 P36888 1/20 0.52
AURKB Q96GD4 1/20 0.52
CLK4 Q9HAZ1 1/20 0.52
MKNK2 Q9HBH9 1/20 0.52
MAPT P10636 3/20 0.50
ALDH1A1 P00352 2/20 0.50
GRM1 Q13255 1/20 0.50
MEN1 O00255 1/20 0.49
NPC1 O15118 1/20 0.49
TP53 P04637 1/20 0.49
MAPK1 P28482 1/20 0.49
RAB9A P51151 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8889590 0.99 EGFR (0.71) EGFRERBB2NPY5RSLC2A1MERTK
SCHEMBL8890861 0.89 NPY5R (0.77) EGFRERBB2NPY5RSLC2A1MERTK
Hydrochloric Acid SCHEMBL8893122 0.89 NPY5R (0.67) EGFRERBB2NPY5RSLC2A1MERTK
Hydrochloric Acid SCHEMBL8899212 0.88 NPY5R (0.76) EGFRERBB2NPY5RSLC2A1MERTK
Hydrochloric Acid SCHEMBL8889878 0.87 NPY5R (0.78) EGFRNPY5RSLC2A1MERTKMAPT
SCHEMBL8899542 0.86 NPY5R (0.69) EGFRERBB2NPY5RSLC2A1MERTK
SCHEMBL8900305 0.86 EGFR (0.69) EGFRERBB2NPY5RSLC2A1MERTK
Hydrochloric Acid SCHEMBL8890550 0.85 NPY5R (0.67) EGFRERBB2NPY5RSLC2A1MERTK
Hydrochloric Acid SCHEMBL8899588 0.85 CHEK2 (0.67) EGFRERBB2NPY5RSLC2A1MERTK
SCHEMBL1387244 0.84 EGFR (1.00) EGFRERBB2ERBB4CHEK2ROS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO claimed